---
version: '1.0'
entity: drug
term: 'hgnc.symbol:'
ordered: false
label: '{entity} is a target of {term}'
source: https://maayanlab.cloud/DrugEnrichr
---
F2		nafamostat	phenindione	ximelagatran	bivalirudin	dabigatran etexilate	cianidanol	sulfaguanidine	argatroban	dibrompropamidine	apixaban	hexamidine	camostat	captopril	quercetin	bortezomib
GNRHR		triptorelin	degarelix	gonadorelin	goserelin	histrelin	abarelix	ganirelix	leuprolide	cetrorelix	nafarelin
AVPR2		tolvaptan	atosiban	carbetocin	desmopressin	quercetin	clotrimazole	itraconazole	lypressin
AVPR1A		tolvaptan	ritonavir	felypressin	saquinavir	atosiban	carbetocin	desmopressin	diethylstilbestrol	lypressin
DHODH		leflunomide	atovaquone	teriflunomide	oxycinchophen	cyclosporine
FKBP1A		everolimus	temsirolimus	sirolimus	tacrolimus	pimecrolimus	cyclosporine	thiabendazole
TACR2		paclitaxel	raloxifene	cefapirin	miconazole	fluphenazine	metergoline	ebastine	vinorelbine	chlorpromazine	clomifene	oxiconazole	ketoconazole	cyclosporine	nelfinavir	saquinavir	suloctidil	diethylstilbestrol	hexachlorophene	clotrimazole	indinavir	sulconazole	terfenadine	docetaxel	ritonavir	amiodarone	haloprogin	danazol	montelukast	lovastatin	astemizole	bithionol	econazole	tamoxifen
ABCB1		irinotecan	paclitaxel	losartan	teniposide	idarubicin	imatinib	amoxapine	epinastine	aliskiren	cyclobenzaprine	saxagliptin	silodosin	daunorubicin	ebastine	meprobamate	megestrol acetate	alfentanil	ketoconazole	donepezil	sertindole	cyclosporine	fexofenadine	omeprazole	nelfinavir	mitoxantrone	azelastine	ketotifen	progesterone	saquinavir	acrivastine	methotrexate	pimozide	desloratadine	lapatinib	dexniguldipine	terfenadine	everolimus	atazanavir	cyproheptadine	propranolol	ritonavir	midazolam	sirolimus	budesonide	vincristine	topotecan	triflupromazine	tamoxifen	bufuralol	tipranavir	verapamil	etravirine	anhydrovinblastine	azithromycin	lopinavir	reserpine	zolpidem	levocabastine	quinine	chlorpromazine	doxazosin	temsirolimus	loratadine	etoposide	nicardipine	mefloquine	aripiprazole	mometasone furoate	diltiazem	quinidine	domperidone	colchicine	clotrimazole	trifluoperazine	indomethacin	haloperidol	mibefradil	udenafil	docetaxel	propafenone	vinblastine	amiodarone	ranolazine	talinolol	quercetin	astemizole	doxorubicin
CYP3A4		nifedipine	amprenavir	zafirlukast	isoniazid	nimodipine	tacrolimus	warfarin	aliskiren	saxagliptin	itraconazole	candesartan cilexetil	mosapride	dapsone	metyrapone	fluconazole	ethambutol	chloramphenicol	oxiconazole	ketoconazole	idebenone	cyclosporine	omeprazole	nelfinavir	voriconazole	pyrazinamide	saquinavir	ergotamine	indinavir	triazolam	sulconazole	atazanavir	ritonavir	vindesine	midazolam	sirolimus	econazole	topotecan	posaconazole	verapamil	dihydroergotamine	cefapirin	maprotiline	miconazole	atorvastatin	aprepitant	vinorelbine	nicardipine	dihydroergocristine	alprazolam	lacidipine	diltiazem	diazepam	bromocriptine	buspirone	colchicine	clotrimazole	cobicistat	mifepristone	troglitazone	mibefradil	docetaxel	amiodarone	nefazodone	cisapride	cyclophosphamide	phenelzine	astemizole	cycloserine	mezlocillin	podofilox	stiripentol
FPR1		oxyphenbutazone	oxaprozin	deoxycholic acid	sulfinpyrazone	phenylbutazone	chenodeoxycholic acid	cyclosporine
ABCC2		irinotecan	mitoxantrone	saquinavir	etravirine	methotrexate	anhydrovinblastine	azithromycin	vinblastine	etoposide	doxorubicin	vincristine	topotecan	cyclosporine
ABCC1		diosmetin	irinotecan	mitoxantrone	saquinavir	verapamil	idarubicin	colchicine	imatinib	etravirine	methotrexate	anhydrovinblastine	benzbromarone	pimozide	sulfinpyrazone	daunorubicin	indomethacin	vinblastine	etoposide	quercetin	doxorubicin	mezlocillin	vincristine	cyclosporine
ABCG2		irinotecan	mitoxantrone	teniposide	verapamil	imatinib	etravirine	methotrexate	gefitinib	maprotiline	reserpine	azathioprine	daunorubicin	lapatinib	novobiocin	etoposide	nicardipine	quercetin	astemizole	doxorubicin	topotecan	cyclosporine
ABCB11		nifedipine	paclitaxel	acitretin	fusidic acid	dicloxacillin	glyburide	clobetasol propionate	rifampicin	rifamycin	troglitazone	pioglitazone	nefazodone	bosentan	praziquantel	erythromycin	rosiglitazone	ticlopidine	cyclosporine
SLCO1B1		rifampicin	rifamycin	repaglinide	cyclosporine	lapatinib
SSTR5		loperamide	somatostatin	lanreotide	pasireotide	octreotide	astemizole
OPRM1		meperidine	levacetylmethadol	raloxifene	naldemedine	levorphanol	alvimopan	hydromorphone	dihydrocodeine	pentazocine	alfentanil	methadyl acetate	naloxone	cyproterone acetate	nelfinavir	saquinavir	disulfiram	diphenoxylate	oxymorphone	pimozide	loperamide	ritonavir	fentanyl	flunarizine	danazol	difenoxin	meptazinol	methadone	bithionol	econazole	tamoxifen	sufentanil	ethinylestradiol	nalfurafine	cinnarizine	tianeptine	butorphanol	cefapirin	miconazole	tramadol	eluxadoline	reserpine	fluphenazine	codeine	buprenorphine	hydrocodone	chlorpromazine	octreotide	nalmefene	dihydroergocristine	morphine	naltrexone	domperidone	diethylstilbestrol	clotrimazole	dextropropoxyphene	mifepristone	naloxegol	haloperidol	levallorphan	amiodarone	tilidine	dezocine	ketobemidone	nalorphine	nalbuphine	oxycodone	anileridine	astemizole	remifentanil
SSTR4		somatostatin	cefonicid	lanreotide	octreotide	cefradine	cefapirin	cefalotin
GSR		methylene blue	nifedipine	carmustine	glutamic acid	menadione	l-lysine
TYR		hexylresorcinol	ascorbic acid	arbutin	kojic acid	mequinol	monobenzone	avobenzone	mimosine
SRC		niclosamide	sunitinib	erlotinib	ponatinib	sorafenib	imatinib	gefitinib	ceritinib	nilotinib	afatinib	dasatinib	crizotinib	ibrutinib	pazopanib	trabectedin	vandetanib	adenosine phosphate	nintedanib	quercetin	bosutinib	rivoceranib
CYP19A1		doconexent	alpha-linolenic acid	anastrozole	exemestane	letrozole	nimesulide	masoprocol	testosterone	oleic acid	androstenedione	clotrimazole	miconazole	testolactone	linoleic acid	formestane	aminoglutethimide	ketoconazole	quercetin	stanolone	icosapent	vorozole
PTGS1		alpha-linolenic acid	diclofenac	dexibuprofen	oxametacin	isoxicam	oxaprozin	acetylsalicylic acid	linoleic acid	mefenamic acid	fenbufen	tolfenamic acid	ipriflavone	valdecoxib	monobenzone	diethylcarbamazine	meclofenamic acid	oxacillin	phenylbutazone	tiaprofenic acid	balsalazide	mesalazine	nimesulide	propofol	celecoxib	parecoxib	tenidap	piroxicam	proquazone	ketorolac	etoricoxib	capsaicin	thalidomide	azapropazone	tolmetin	loxoprofen	suprofen	bromfenac	flufenamic acid	tamoxifen	nabumetone	flurbiprofen	cianidanol	ibuprofen	alclofenac	eugenol	indobufen	acemetacin	aminosalicylic acid	lumiracoxib	fenoprofen	rofecoxib	ketoprofen	pirprofen	dexketoprofen	niflumic acid	captopril	clomifene	zomepirac	mercaptopurine	tenoxicam	diflunisal	carprofen	nepafenac	bismuth subsalicylate	oxyphenbutazone	tioguanine	diethylstilbestrol	etodolac	phenacetin	indomethacin	naproxen	meloxicam	felbinac	sulfasalazine	ticlopidine	mezlocillin	aminophenazone	floctafenine
PPARG		balsalazide	alpha-linolenic acid	diclofenac	telmisartan	bezafibrate	mesalazine	oleic acid	stearic acid	saroglitazar	troglitazone	indomethacin	linoleic acid	gamolenic acid	bexarotene	pioglitazone	lauric acid	rosiglitazone	fenofibrate	mezlocillin	lobeglitazone	icosapent
PPARA		alpha-linolenic acid	bezafibrate	oleic acid	stearic acid	fenofibric acid	saroglitazar	linoleic acid	gamolenic acid	clofibrate	gemfibrozil	pioglitazone	ciprofibrate	lauric acid	rosiglitazone	fenofibrate	lobeglitazone	icosapent
PPARD		gamolenic acid	alpha-linolenic acid	bezafibrate	oleic acid	stearic acid	lauric acid	rosiglitazone	tretinoin	icosapent	linoleic acid
F3		gamolenic acid	alpha-linolenic acid	oleic acid	icosapent	linoleic acid
VDR		calcipotriol	calcitriol	ergocalciferol	paricalcitol	eldecalcitol	calcifediol	cholecalciferol	doxercalciferol	alfacalcidol	dihydrotachysterol	tacalcitol
GRIA3		topiramate	glutamic acid	perampanel	cyclothiazide	ketamine
ADORA3		nifedipine	zafirlukast	theophylline	nimodipine	mitotane	benzbromarone	candesartan cilexetil	ebastine	prazosin	oxiconazole	fenofibrate	naloxone	felodipine	glutamic acid	nelfinavir	celecoxib	disulfiram	suloctidil	hexachlorophene	tretinoin	sulconazole	mepyramine	dexniguldipine	nitrendipine	caffeine	flunarizine	danazol	istradefylline	bithionol	econazole	rabeprazole	tamoxifen	isotretinoin	estradiol benzoate	baclofen	ethinylestradiol	imipramine	stanozolol	miconazole	ketanserin	yohimbine	adenosine	fluphenazine	nisoldipine	protriptyline	clomifene	clozapine	nicardipine	enprofylline	lacidipine	pirenzepine	diazepam	tioguanine	hydroxyprogesterone caproate	diethylstilbestrol	clotrimazole	diiodohydroxyquinoline	troglitazone	amiodarone	atenolol	haloprogin	montelukast	quercetin	astemizole	mezlocillin
GRIA4		topiramate	glutamic acid	perampanel	cyclothiazide	ketamine
GRIA2		topiramate	glutamic acid	perampanel	cyclothiazide	ketamine
GRIA1		topiramate	glutamic acid	perampanel	cyclothiazide	ketamine
TYMS		folic acid	pemetrexed	floxuridine	gemcitabine	capecitabine	doxifluridine	levomefolic acid	phenolphthalein	raltitrexed	fluorouracil	methotrexate	leucovorin
GLRA1		nifedipine	telmisartan	dutasteride	isoflurane	risperidone	enflurane	fluspirilene	desflurane	colchicine	regorafenib	ethanol	pimozide	tropisetron	methohexital	sulindac	cinacalcet	adapalene	cholecalciferol	dronabinol	sevoflurane	halothane	astemizole	mefloquine	methoxyflurane
MAOA		nabumetone	pargyline	iproniazid	nomifensine	isocarboxazid	pheniprazine	amiloride	selegiline	debrisoquine	safinamide	pioglitazone	menadione	pentamidine	rosiglitazone	ethynodiol diacetate	tranylcypromine	methoxsalen	toloxatone	phenmetrazine	proparacaine	trioxsalen	chloroxylenol	leflunomide	disulfiram	bergapten	troglitazone	dextroamphetamine	methylene blue	linezolid	rasagiline	primaquine	tetracaine	fentanyl	mebanazine	phenelzine	quercetin	guanabenz	moclobemide	pirlindole
MAOB		pargyline	iproniazid	isocarboxazid	pheniprazine	selegiline	debrisoquine	safinamide	pioglitazone	cyclizine	menadione	zonisamide	rosiglitazone	donepezil	tranylcypromine	toloxatone	troglitazone	methylene blue	linezolid	rasagiline	primaquine	fentanyl	hymecromone	mebanazine	phenelzine	quercetin	moclobemide
IDO1		isoconazole	menadione	sertaconazole	mitomycin	oxiconazole	ketoconazole	phenelzine	dichlorophen	miconazole	econazole	sulconazole	bifonazole
ACE		omapatrilat	telmisartan	losartan	temocapril	moexipril	enalapril	zofenopril	benazepril	cilazapril	racecadotril	enalaprilat	fosinopril	perindopril	lisinopril	proline	quinapril	ramipril	captopril	imidapril	delapril	spirapril	trandolapril
XDH		adenine	tioguanine	topiroxostat	azapropazone	rutin	febuxostat	quercetin	allopurinol
HMGCR		bezafibrate	cerivastatin	fluvastatin	pitavastatin	cisapride	pravastatin	meglutol	simvastatin	lovastatin	rosuvastatin	atorvastatin
SIGMAR1		zidovudine	nepinalone	fluvoxamine	terconazole	amantadine	mosapride	thiethylperazine	pentazocine	donepezil	ifenprodil	risperidone	casopitant	trihexyphenidyl	pentoxyverine	promethazine	fluoxetine	mazindol	propranolol	flunarizine	tamoxifen	amitriptyline	lamotrigine	testosterone	imipramine	trazodone	cinnarizine	methysergide	buflomedil	perhexiline	trifluperidol	paroxetine	chlorpromazine	clomifene	tolperisone	promazine	eperisone	bromperidol	clomipramine	labetalol	benperidol	valethamate	metamfetamine	buspirone	benzatropine	butenafine	tetracaine	iloperidone	propafenone	caramiphen	clemastine	ticlopidine	astemizole	sertraline	dicyclomine	molindone	raloxifene	dextromethorphan	remoxipride	diphenidol	prochlorperazine	proparacaine	etilamfetamine	blonanserin	progesterone	quetiapine	suloctidil	pimozide	mepyramine	loperamide	dobutamine	citalopram	econazole	terbinafine	thioridazine	cefapirin	levobunolol	bromhexine	ketanserin	fluphenazine	oxybutynin	flupentixol	clozapine	doxepin	opipramol	cocaine	trifluoperazine	mifepristone	haloperidol	phentolamine	phencyclidine	amiodarone	cisapride	dexfenfluramine	nalorphine	dexchlorpheniramine	naftifine	pramocaine
SLC6A3		levomilnacipran	methylphenidate	dicloxacillin	mitotane	nomifensine	phenylpropanolamine	fluvoxamine	terconazole	metergoline	ebastine	sibutramine	cyclizine	duloxetine	oxiconazole	ketoconazole	fenofibrate	dosulepin	tranylcypromine	nelfinavir	norepinephrine	diethylpropion	celecoxib	disulfiram	lisdexamfetamine	zotepine	sulconazole	desipramine	fluoxetine	terfenadine	mazindol	flunarizine	tamoxifen	amitriptyline	pemoline	imipramine	trazodone	modafinil	cinnarizine	miconazole	paroxetine	phendimetrazine	chlorpromazine	clomifene	armodafinil	dopamine	aripiprazole	clomipramine	labetalol	diphenhydramine	metamfetamine	amlodipine	benzatropine	clotrimazole	iloperidone	propafenone	haloprogin	nefazodone	iprindole	montelukast	clemastine	phenelzine	astemizole	estradiol	reboxetine	sertraline	meperidine	amoxapine	raloxifene	mianserin	phentermine	chlorphentermine	bupropion	prochlorperazine	nimesulide	leflunomide	saquinavir	dexmethylphenidate	suloctidil	desloratadine	dextroamphetamine	mepyramine	venlafaxine	danazol	viloxazine	dobutamine	citalopram	bithionol	econazole	milnacipran	nortriptyline	ethinylestradiol	ziprasidone	trovafloxacin	thioridazine	amphetamine	maprotiline	fluphenazine	diphenylpyraline	chlorpheniramine	protriptyline	bisacodyl	doxazosin	oxybutynin	pentamidine	asenapine	nefopam	phenmetrazine	hydroxyprogesterone caproate	carvedilol	cocaine	diethylstilbestrol	trimipramine	atomoxetine	amiodarone	methapyrilene	brexpiprazole	lovastatin	dexchlorpheniramine
SLC6A4		levomilnacipran	methylphenidate	desvenlafaxine	mitotane	cyclobenzaprine	nomifensine	carbamazepine	fluvoxamine	terconazole	metergoline	mosapride	ebastine	sibutramine	duloxetine	oxiconazole	ketoconazole	donepezil	tibolone	dosulepin	vilazodone	ethylestrenol	risperidone	celecoxib	etoperidone	zotepine	sulconazole	ambroxol	desipramine	olanzapine	promethazine	fluoxetine	primaquine	mazindol	dapoxetine	propranolol	flunarizine	orphenadrine	escitalopram	tamoxifen	amitriptyline	imipramine	trazodone	verapamil	cinnarizine	miconazole	levonorgestrel	paroxetine	estriol	chlorpromazine	clomifene	promazine	aripiprazole	clomipramine	diphenhydramine	metamfetamine	benzatropine	clotrimazole	thiothixene	butenafine	haloprogin	nefazodone	iprindole	astemizole	estradiol	reboxetine	sertraline	imatinib	amoxapine	raloxifene	dextromethorphan	mianserin	norethisterone	chlorphentermine	bupropion	prochlorperazine	vortioxetine	clopidogrel	suloctidil	hexachlorophene	desloratadine	dextroamphetamine	mepyramine	loperamide	venlafaxine	ofloxacin	cyproheptadine	danazol	viloxazine	dobutamine	citalopram	econazole	fenfluramine	milnacipran	estradiol benzoate	nortriptyline	ethinylestradiol	ziprasidone	thioridazine	amphetamine	maprotiline	tramadol	levobunolol	bromhexine	reserpine	mestranol	tropisetron	fluphenazine	chlorpheniramine	protriptyline	doxazosin	lorcaserin	zimelidine	clozapine	doxepin	nefopam	carvedilol	cocaine	domperidone	diethylstilbestrol	trimipramine	atomoxetine	haloperidol	estrone	amiodarone	lofepramine	cisapride	dexfenfluramine	methapyrilene	brexpiprazole	dexchlorpheniramine	paliperidone
CYP1A2		nifedipine	nabumetone	altretamine	modafinil	thioridazine	fluvoxamine	mosapride	nisoldipine	paroxetine	armodafinil	thiabendazole	flutamide	methoxsalen	omeprazole	prochlorperazine	leflunomide	pefloxacin	disulfiram	hexachlorophene	tenidap	sulconazole	alosetron	artemisinin	primaquine	atazanavir	propafenone	propranolol	capsaicin	econazole	stiripentol
SLC6A2		levomilnacipran	methylphenidate	pseudoephedrine	desvenlafaxine	mitotane	cyclobenzaprine	nomifensine	phenylpropanolamine	fluvoxamine	terconazole	metergoline	ebastine	sibutramine	guanadrel	valdecoxib	duloxetine	loxapine	oxiconazole	ketoconazole	fenofibrate	dosulepin	tranylcypromine	nelfinavir	ethylestrenol	propofol	riluzole	diethylpropion	celecoxib	disulfiram	lisdexamfetamine	zotepine	sulconazole	desipramine	promethazine	fluoxetine	terfenadine	mazindol	flunarizine	orphenadrine	escitalopram	tamoxifen	amitriptyline	nabumetone	imipramine	trazodone	cinnarizine	miconazole	perhexiline	paroxetine	phendimetrazine	chlorpromazine	clomifene	dopamine	promazine	aripiprazole	clomipramine	labetalol	diphenhydramine	tacrine	metamfetamine	benzatropine	clotrimazole	butenafine	alfacalcidol	iloperidone	propafenone	guanethidine	haloprogin	nefazodone	iprindole	montelukast	clemastine	astemizole	reboxetine	sertraline	amoxapine	raloxifene	candesartan cilexetil	mianserin	ipriflavone	monobenzone	phentermine	bupropion	benzphetamine	mitoxantrone	prochlorperazine	leflunomide	dexmethylphenidate	quetiapine	suloctidil	desloratadine	dextroamphetamine	venlafaxine	cyproheptadine	danazol	viloxazine	dobutamine	citalopram	bithionol	econazole	milnacipran	estradiol benzoate	mirtazapine	nortriptyline	ethinylestradiol	ziprasidone	terbinafine	thioridazine	amphetamine	bethanidine	epinephrine	maprotiline	tramadol	mestranol	fluphenazine	chlorpheniramine	protriptyline	quinacrine	oxybutynin	pentamidine	zimelidine	clozapine	doxepin	lacidipine	nefopam	phenmetrazine	carvedilol	cocaine	domperidone	diethylstilbestrol	trimipramine	atomoxetine	haloperidol	amiodarone	lofepramine	methapyrilene	brexpiprazole	lovastatin	dexchlorpheniramine
AGTR1		telmisartan	irbesartan	losartan	eprosartan	fimasartan	saralasin	valsartan	azilsartan medoxomil	tasosartan	candesartan cilexetil
ALOX5		balsalazide	mesalazine	masoprocol	mizolastine	ibuprofen	zileuton	chloroxine	hexylresorcinol	benoxaprofen	montelukast	quercetin	sulfasalazine	diethylcarbamazine	mezlocillin	meclofenamic acid
AR		bicalutamide	drostanolone propionate	dexamethasone	exemestane	ethinylestradiol	masoprocol	testosterone	stanozolol	flucloxacillin	oxymetholone	testosterone enanthate	prednisolone	norethisterone	tolfenamic acid	medroxyprogesterone acetate	tibolone	meclofenamic acid	cyproterone acetate	flutamide	methyltestosterone	testosterone cypionate	ethylestrenol	progesterone	oxandrolone	testosterone undecanoate	mifepristone	nandrolone decanoate	indomethacin	spironolactone	androstenediol	fluoxymesterone	testosterone propionate	nandrolone phenpropionate	danazol	nilutamide	drospirenone	flufenamic acid	nandrolone	stanolone	tiratricol	estradiol	enzalutamide
IGF1R		sunitinib	crizotinib	masoprocol	nintedanib	quercetin	ceritinib
ESR1		estradiol benzoate	ethinylestradiol	estradiol valerate	masoprocol	stanozolol	etonogestrel	oxymetholone	raloxifene	mestranol	levonorgestrel	estriol	norethisterone	bazedoxifene	clomifene	estradiol acetate	medroxyprogesterone acetate	toremifene	ethynodiol diacetate	tibolone	chlorotrianisene	estradiol cypionate	ethylestrenol	fulvestrant	progesterone	diethylstilbestrol	hexachlorophene	moxestrol	gossypol	lasofoxifene	ospemifene	mifepristone	quinestrol	androstenediol	estrone	nandrolone phenpropionate	ethyl hydroxybenzoate	danazol	hexestrol	bithionol	estradiol	tamoxifen
TTR		nifedipine	diclofenac	masoprocol	tafamidis	nitrendipine	gemfibrozil	niflumic acid	tolfenamic acid	aceclofenac	diflunisal	flufenamic acid	levothyroxine	meclofenamic acid
NR3C1		dexamethasone	ciclesonide	amcinonide	megestrol acetate	prednisolone	betamethasone	triamcinolone	norethisterone	medrysone	hydrocortisone	meprednisone	hydrocortisone valerate	beclomethasone dipropionate	hydrocortamate	cyproterone acetate	methyltestosterone	loteprednol etabonate	hydrocortisone cypionate	fluocinonide	clobetasol propionate	progesterone	flurandrenolide	spironolactone	budesonide	danazol	prednisolone tebutate	hydrocortisone butyrate	fluocinolone acetonide	flunisolide	fluticasone furoate	estradiol benzoate	ethinylestradiol	testosterone	hydrocortisone acetate	methylprednisolone	levonorgestrel	cortisone acetate	rimexolone	estriol	cortivazol	fluorometholone	fluticasone propionate	prednicarbate	medroxyprogesterone acetate	prednisone	fluprednisolone	mometasone furoate	hydroxyprogesterone caproate	methylprednisolone hemisuccinate	prednisolone acetate	eplerenone	diethylstilbestrol	clotrimazole	difluprednate	mifepristone	hydrocortisone probutate	desonide	halcinonide	dexamethasone acetate	desoximetasone	podofilox	estradiol
TAAR1		histamine	octopamine	tolazoline	metamfetamine	amphetamine	tyramine	dopamine	hydroxyamphetamine	levmetamfetamine	dextroamphetamine
ADRA1A		piribedil	pseudoephedrine	clonidine	epinastine	phenylpropanolamine	nylidrin	mephentermine	guanadrel	thiethylperazine	loxapine	prazosin	apomorphine	dosulepin	sertindole	vilazodone	brimonidine	norepinephrine	risperidone	zotepine	desipramine	olanzapine	promethazine	fluoxetine	terfenadine	rilmenidine	escitalopram	amitriptyline	imipramine	trazodone	cabergoline	dihydroergotamine	buflomedil	tolazoline	chlorpromazine	xylometazoline	promazine	aripiprazole	bromperidol	clomipramine	diazepam	midodrine	bromocriptine	bunazosin	lisuride	buspirone	amlodipine	medetomidine	thiothixene	iloperidone	guanethidine	nefazodone	phenylephrine	urapidil	pergolide	sertraline	molindone	perphenazine	methoxamine	oxymetazoline	silodosin	mianserin	alfuzosin	terazosin	tamsulosin	bupropion	zuclopenthixol	benzphetamine	dexmedetomidine	prochlorperazine	azelastine	blonanserin	ergotamine	quetiapine	pimozide	terguride	dextroamphetamine	dexniguldipine	metaraminol	naftopidil	cyproheptadine	phenoxybenzamine	droxidopa	fenfluramine	mirtazapine	nortriptyline	tetryzoline	ziprasidone	thioridazine	amphetamine	epinephrine	maprotiline	ketanserin	yohimbine	fluphenazine	indoramin	doxazosin	flupentixol	clozapine	asenapine	dihydroergocristine	doxepin	apraclonidine	melperone	carvedilol	cocaine	domperidone	trifluoperazine	haloperidol	phentolamine	lofepramine	dexfenfluramine	brexpiprazole	fenoldopam	dapiprazole	paliperidone
ADRA2A		methylphenidate	piribedil	pseudoephedrine	mitotane	clonidine	epinastine	methyldopa	phenylpropanolamine	tetrabenazine	terconazole	metergoline	mosapride	ebastine	gabapentin	cyclizine	loxapine	prazosin	oxiconazole	ketoconazole	apomorphine	sertindole	vilazodone	brimonidine	naphazoline	tramazoline	tizanidine	norepinephrine	risperidone	ketotifen	ergometrine	tiapride	disulfiram	zotepine	sulconazole	desipramine	olanzapine	promethazine	fluoxetine	amisulpride	dipivefrin	rilmenidine	flunarizine	orphenadrine	tamoxifen	amitriptyline	ropinirole	trazodone	verapamil	cinnarizine	methysergide	benzquinamide	cabergoline	dihydroergotamine	miconazole	buflomedil	pipamperone	moxonidine	tolazoline	chlorpromazine	clomifene	xylometazoline	promazine	aripiprazole	clomipramine	droperidol	bromocriptine	lisuride	metamfetamine	amlodipine	benzatropine	clotrimazole	medetomidine	thiothixene	butenafine	iloperidone	guanethidine	haloprogin	montelukast	phenylephrine	vancomycin	clemastine	ticlopidine	astemizole	guanabenz	pergolide	sertraline	lofexidine	molindone	perphenazine	oxymetazoline	amoxapine	raloxifene	mianserin	selegiline	terazosin	lurasidone	pramipexole	tamsulosin	benzphetamine	dexmedetomidine	prochlorperazine	ergotamine	quetiapine	suloctidil	hexachlorophene	pimozide	terguride	dextroamphetamine	mepyramine	dexniguldipine	cyproheptadine	metoclopramide	danazol	phenoxybenzamine	droxidopa	bithionol	econazole	fenfluramine	sulpiride	mirtazapine	nortriptyline	tetryzoline	ziprasidone	terbinafine	thioridazine	amphetamine	epinephrine	maprotiline	ketanserin	yohimbine	fluphenazine	quinacrine	indoramin	emetine	doxazosin	pentamidine	clozapine	asenapine	dihydroergocristine	doxepin	apraclonidine	melperone	levonordefrin	fluspirilene	carvedilol	domperidone	rutin	diethylstilbestrol	trifluoperazine	methylergometrine	haloperidol	phentolamine	guanfacine	amiodarone	cisapride	dexfenfluramine	methapyrilene	brexpiprazole	dexchlorpheniramine	paliperidone
CCKBR		proglumide	sincalide	iloperidone	pentagastrin	chlordiazepoxide
CHRNA4		hexamethonium	mecamylamine	nicotine	pipecuronium	varenicline	alcuronium	ondansetron	granisetron	acetylcholine	tropisetron
CHRNB2		hexamethonium	mecamylamine	nicotine	pipecuronium	varenicline	metocurine	ondansetron	granisetron	acetylcholine	bupropion	tropisetron	methohexital
CHRNA1		procaine	nicotine	pipecuronium	metocurine	decamethonium	gallamine	succinylcholine	lidocaine	tropisetron	mecamylamine	varenicline	alcuronium	mivacurium
CHRNB1		procaine	nicotine	pipecuronium	varenicline	alcuronium	metocurine	mivacurium	decamethonium	succinylcholine	lidocaine	tropisetron
CHRND		procaine	nicotine	pipecuronium	varenicline	alcuronium	metocurine	mivacurium	decamethonium	succinylcholine	lidocaine	tropisetron
CHRNG		nicotine	varenicline	decamethonium	succinylcholine	tropisetron
HTR3A		procaine	mirtazapine	nicotine	lamotrigine	ziprasidone	memantine	ramosetron	cyamemazine	granisetron	amoxapine	tyramine	tropisetron	mianserin	mosapride	dolasetron	chlorpromazine	ondansetron	clozapine	loxapine	sumatriptan	aripiprazole	asenapine	octopamine	diltiazem	bupivacaine	vortioxetine	cocaine	prucalopride	thiothixene	tegaserod	zotepine	lidocaine	olanzapine	alosetron	levobupivacaine	metoclopramide	cisapride	astemizole
HTR3B		nicotine	metoclopramide	ondansetron	cocaine	cisapride	granisetron	tropisetron
CHRNA3		pentolinium	mecamylamine	nicotine	varenicline	granisetron	trimethaphan	bupropion	tropisetron
CHRNB4		pentolinium	hexamethonium	mecamylamine	nicotine	pipecuronium	varenicline	alcuronium	trimethaphan	carbamazepine	bupropion
KCND3		sibutramine	guanidine	nicotine	levobupivacaine	bupivacaine	dalfampridine	amifampridine
CHRNA7		mecamylamine	nicotine	varenicline	alcuronium	naltrexone	acetylcholine	trimethaphan	bupropion	tropisetron
TRPA1		thymol	nicotine	propyphenazone	antipyrine	dronabinol	apomorphine
CHRNA2		biperiden	mecamylamine	nicotine	pipecuronium	alcuronium	metocurine	mivacurium	carbamazepine	methohexital
CHRM3		dicloxacillin	anisotropine methylbromide	butylscopolamine	imidafenacin	cyclobenzaprine	terconazole	ebastine	thiethylperazine	cyclizine	pridinol	acetylcholine	loxapine	oxiconazole	dosulepin	sertindole	pilocarpine	risperidone	tridihexethyl	ketotifen	xanomeline	trihexyphenidyl	hexocyclium	zotepine	sulconazole	desipramine	olanzapine	promethazine	fluoxetine	aceclidine	flunarizine	hyoscyamine	methantheline	orphenadrine	tamoxifen	amitriptyline	atropine	oxyphencyclimine	imipramine	cyamemazine	cinnarizine	methysergide	miconazole	darifenacin	perhexiline	paroxetine	clidinium	alcuronium	chlorprothixene	chlorpromazine	clomifene	methacholine	promazine	mesoridazine	aripiprazole	bromperidol	clomipramine	diphenhydramine	procyclidine	valethamate	benzatropine	clotrimazole	thiothixene	montelukast	clemastine	astemizole	sertraline	dicyclomine	molindone	biperiden	perphenazine	cyclopentolate	amoxapine	mianserin	disopyramide	isopropamide	bethanechol	dimetindene	diphenidol	prochlorperazine	vinburnine	quetiapine	suloctidil	ipratropium	pimozide	desloratadine	cyproheptadine	carbenicillin	danazol	mepenzolate	fesoterodine	econazole	fenfluramine	scopolamine	nortriptyline	propantheline	ziprasidone	oxyphenonium	thioridazine	maprotiline	methscopolamine	fluphenazine	protriptyline	quinacrine	tolterodine	oxybutynin	clozapine	asenapine	doxepin	tiotropium	cevimeline	pirenzepine	solifenacin	homatropine	vincamine	tropicamide	diethylstilbestrol	trifluoperazine	haloperidol	amiodarone	lofepramine	propiomazine	mequitazine	dexfenfluramine	dexchlorpheniramine
CHRM1		dicloxacillin	anisotropine methylbromide	butylscopolamine	imidafenacin	cyclobenzaprine	phenylpropanolamine	terconazole	ebastine	thiethylperazine	cyclizine	pridinol	acetylcholine	loxapine	oxiconazole	dosulepin	pilocarpine	risperidone	tridihexethyl	ketotifen	xanomeline	trihexyphenidyl	hexocyclium	zotepine	sulconazole	desipramine	olanzapine	pentoxyverine	promethazine	fluoxetine	terfenadine	aceclidine	flunarizine	hyoscyamine	methantheline	orphenadrine	escitalopram	tamoxifen	amitriptyline	atropine	linagliptin	oxyphencyclimine	imipramine	cyamemazine	cinnarizine	methysergide	pyrimethamine	miconazole	darifenacin	perhexiline	paroxetine	clidinium	alcuronium	chlorprothixene	chlorpromazine	clomifene	methacholine	promazine	mesoridazine	aripiprazole	bromperidol	clomipramine	diphenhydramine	procyclidine	valethamate	cycrimine	gallamine	benzatropine	clotrimazole	thiothixene	iloperidone	montelukast	oxatomide	clemastine	astemizole	doxorubicin	mebhydrolin	sertraline	dicyclomine	biperiden	amoxapine	mianserin	disopyramide	isopropamide	bethanechol	dimetindene	diphenidol	minaprine	mitoxantrone	prochlorperazine	vinburnine	ergotamine	quetiapine	suloctidil	ipratropium	desloratadine	ofloxacin	cyproheptadine	carbenicillin	metoclopramide	mepenzolate	metixene	fesoterodine	citalopram	econazole	fenfluramine	scopolamine	mirtazapine	nortriptyline	propantheline	ziprasidone	oxyphenonium	thioridazine	maprotiline	methscopolamine	fluphenazine	diphenylpyraline	protriptyline	quinacrine	tolterodine	oxybutynin	clozapine	asenapine	doxepin	tiotropium	cevimeline	pirenzepine	solifenacin	homatropine	vincamine	pizotifen	tropicamide	diethylstilbestrol	profenamine	haloperidol	amiodarone	lofepramine	propiomazine	mequitazine	dexfenfluramine	methapyrilene	dexchlorpheniramine
CHRM5		dicyclomine	biperiden	oxymetazoline	amoxapine	terconazole	mianserin	ebastine	thiethylperazine	cyclizine	pridinol	acetylcholine	dimetindene	loxapine	diphenidol	dosulepin	pilocarpine	nelfinavir	prochlorperazine	ketotifen	xanomeline	quetiapine	suloctidil	trihexyphenidyl	hexocyclium	zotepine	ipratropium	sulconazole	desipramine	desloratadine	olanzapine	promethazine	fluoxetine	aceclidine	cyproheptadine	flunarizine	hyoscyamine	methantheline	fesoterodine	orphenadrine	scopolamine	tamoxifen	amitriptyline	atropine	nortriptyline	ziprasidone	imipramine	cyamemazine	cinnarizine	thioridazine	maprotiline	methscopolamine	darifenacin	perhexiline	tropisetron	fluphenazine	protriptyline	quinacrine	paroxetine	tolterodine	chlorprothixene	chlorpromazine	oxybutynin	clomifene	pentamidine	clozapine	promazine	mesoridazine	aripiprazole	asenapine	bromperidol	clomipramine	diphenhydramine	doxepin	procyclidine	tiotropium	cevimeline	pirenzepine	solifenacin	droperidol	homatropine	valethamate	rutin	tropicamide	benzatropine	thiothixene	haloperidol	amiodarone	lofepramine	propiomazine	mequitazine	methapyrilene	clemastine	astemizole	dexchlorpheniramine	sertraline
CHRM4		butylscopolamine	terconazole	ebastine	thiethylperazine	cyclizine	pridinol	acetylcholine	loxapine	dosulepin	pilocarpine	risperidone	ketotifen	xanomeline	trihexyphenidyl	hexocyclium	zotepine	sulconazole	desipramine	olanzapine	promethazine	fluoxetine	aceclidine	flunarizine	hyoscyamine	methantheline	orphenadrine	tamoxifen	amitriptyline	atropine	imipramine	cyamemazine	cinnarizine	miconazole	darifenacin	perhexiline	paroxetine	alcuronium	chlorprothixene	chlorpromazine	clomifene	methacholine	promazine	mesoridazine	aripiprazole	bromperidol	clomipramine	diphenhydramine	procyclidine	droperidol	valethamate	benzatropine	clotrimazole	thiothixene	iloperidone	clemastine	astemizole	sertraline	dicyclomine	irinotecan	biperiden	oxymetazoline	amoxapine	mianserin	bethanechol	dimetindene	diphenidol	mitoxantrone	prochlorperazine	vinburnine	quetiapine	suloctidil	ipratropium	desloratadine	cyproheptadine	fesoterodine	econazole	fenfluramine	scopolamine	nortriptyline	propantheline	ziprasidone	thioridazine	maprotiline	methscopolamine	fluphenazine	protriptyline	quinacrine	tolterodine	oxybutynin	pentamidine	clozapine	doxepin	tiotropium	cevimeline	melperone	pirenzepine	solifenacin	homatropine	vincamine	tropicamide	amiodarone	lofepramine	propiomazine	mequitazine	dexfenfluramine	dexchlorpheniramine
CHRM2		dicloxacillin	butylscopolamine	cyclobenzaprine	terconazole	ebastine	thiethylperazine	cyclizine	pridinol	acetylcholine	loxapine	ketoconazole	dosulepin	pilocarpine	dexetimide	ethylestrenol	risperidone	ketotifen	xanomeline	trihexyphenidyl	hexocyclium	zotepine	desipramine	olanzapine	pentoxyverine	promethazine	fluoxetine	procainamide	aceclidine	hyoscyamine	methantheline	orphenadrine	tamoxifen	amitriptyline	atropine	imipramine	cyamemazine	methysergide	miconazole	darifenacin	paroxetine	alcuronium	chlorprothixene	chlorpromazine	clomifene	methacholine	promazine	eperisone	mesoridazine	aripiprazole	bromperidol	clomipramine	diphenhydramine	procyclidine	quinidine	valethamate	gallamine	benzatropine	clotrimazole	thiothixene	iloperidone	clemastine	astemizole	sertraline	dicyclomine	biperiden	amoxapine	mianserin	disopyramide	bethanechol	dimetindene	diphenidol	mitoxantrone	prochlorperazine	vinburnine	ergotamine	quetiapine	ipratropium	desloratadine	cyproheptadine	mepenzolate	fesoterodine	econazole	fenfluramine	scopolamine	mirtazapine	nortriptyline	propantheline	ziprasidone	decamethonium	thioridazine	maprotiline	methscopolamine	fluphenazine	protriptyline	quinacrine	tolterodine	oxybutynin	pentamidine	clozapine	asenapine	doxepin	tiotropium	cevimeline	melperone	pirenzepine	solifenacin	homatropine	vincamine	tropicamide	amiodarone	lofepramine	propiomazine	hydroxychloroquine	mequitazine	dexfenfluramine	methapyrilene	dexchlorpheniramine
GABRA1		loprazolam	zopiclone	prazepam	amoxapine	lorazepam	secobarbital	carbamazepine	acamprosate	eltanolone	methylphenobarbital	flunitrazepam	meprobamate	hexobarbital	pentobarbital	quazepam	methoxyflurane	butalbital	triclofos	isoflurane	propofol	triazolam	butabarbital	chlordiazepoxide	lindane	bromazepam	nitrazepam	clonazepam	midazolam	thiopental	liothyronine	progabide	flumazenil	nordazepam	primidone	zaleplon	methyprylon	temazepam	fospropofol	norfloxacin	ethchlorvynol	etizolam	metharbital	estazolam	methohexital	zolpidem	phenobarbital	glutethimide	thiamylal	delorazepam	sevoflurane	etomidate	thiocolchicoside	alfaxalone	adinazolam	alprazolam	talbutal	oxazepam	diazepam	eszopiclone	desflurane	flurazepam	halazepam	topiramate	clobazam	methaqualone	halothane
GABRB3		zaleplon	loprazolam	zopiclone	methyprylon	fospropofol	ethchlorvynol	etizolam	lorazepam	metharbital	estazolam	acamprosate	methohexital	methylphenobarbital	flunitrazepam	meprobamate	zolpidem	glutethimide	hexobarbital	pentobarbital	thiamylal	delorazepam	sevoflurane	methoxyflurane	adinazolam	alprazolam	talbutal	butalbital	triclofos	isoflurane	oxazepam	diazepam	propofol	desflurane	triazolam	chlordiazepoxide	halazepam	lindane	methaqualone	clonazepam	midazolam	halothane	liothyronine	progabide	flumazenil
GABRG2		loprazolam	zopiclone	prazepam	amoxapine	lorazepam	secobarbital	carbamazepine	acamprosate	eltanolone	methylphenobarbital	flunitrazepam	meprobamate	hexobarbital	pentobarbital	quazepam	methoxyflurane	butalbital	triclofos	isoflurane	propofol	triazolam	butabarbital	chlordiazepoxide	lindane	bromazepam	nitrazepam	clonazepam	midazolam	thiopental	liothyronine	progabide	flumazenil	nordazepam	primidone	zaleplon	methyprylon	temazepam	fospropofol	ethchlorvynol	etizolam	metharbital	estazolam	methohexital	zolpidem	phenobarbital	glutethimide	thiamylal	delorazepam	sevoflurane	etomidate	thiocolchicoside	alfaxalone	adinazolam	alprazolam	talbutal	oxazepam	diazepam	eszopiclone	desflurane	flurazepam	halazepam	topiramate	clobazam	methaqualone	halothane
ADRB1		nadolol	timolol	betaxolol	practolol	arbutamine	indacaterol	sotalol	prenalterol	xamoterol	sertindole	norepinephrine	penbutolol	etilefrine	risperidone	vortioxetine	ergotamine	quetiapine	formoterol	zotepine	bupranolol	terguride	olanzapine	fluoxetine	propranolol	acebutolol	alprenolol	dobutamine	droxidopa	oxprenolol	econazole	fenfluramine	levobetaxolol	tamoxifen	tretoquinol	ziprasidone	bufuralol	landiolol	epinephrine	miconazole	levobunolol	darifenacin	salbutamol	clenbuterol	nebivolol	pipamperone	paroxetine	metoprolol	pindolol	celiprolol	clozapine	carteolol	arformoterol	dopamine	metipranolol	aripiprazole	asenapine	esmolol	labetalol	bromocriptine	fluspirilene	carvedilol	lisuride	diethylstilbestrol	clotrimazole	olodaterol	bopindolol	propafenone	amiodarone	atenolol	dexfenfluramine	talinolol	vilanterol	brexpiprazole	salmeterol	astemizole	bevantolol	bisoprolol	paliperidone	isoprenaline	lysergic acid diethylamide
CYP2C19		bicalutamide	nortriptyline	nimodipine	stanozolol	modafinil	thioridazine	miconazole	lansoprazole	noscapine	mosapride	fluconazole	oxybutynin	armodafinil	loratadine	medroxyprogesterone acetate	oxiconazole	tibolone	bupropion	dihydroergocristine	finasteride	idebenone	omeprazole	lacidipine	voriconazole	ethylestrenol	tolnaftate	tropicamide	hexachlorophene	clotrimazole	thiamphenicol	papaverine	spironolactone	sulconazole	nitrendipine	sirolimus	clemastine	phenelzine	ticlopidine	bortezomib	econazole	podofilox	stiripentol	sertraline
LCK		axitinib	sunitinib	erlotinib	imatinib	gefitinib	tirilazad	ceritinib	afatinib	crizotinib	pazopanib	acetic acid	vandetanib	nelfinavir	sorafenib	ergotamine	ruboxistaurin	hexachlorophene	tofacitinib	diiodohydroxyquinoline	nilotinib	dasatinib	ibrutinib	levodopa	carbidopa	dobutamine	nintedanib	quercetin	astemizole	doxorubicin	bithionol	bosutinib	tamoxifen
FYN		paclitaxel	imatinib	methyldopa	raloxifene	itraconazole	tirilazad	terconazole	ebastine	crizotinib	nelfinavir	mitoxantrone	prochlorperazine	ergotamine	suloctidil	hexachlorophene	sulconazole	nilotinib	terfenadine	levodopa	dobutamine	econazole	tamoxifen	estradiol benzoate	sunitinib	thioridazine	miconazole	perhexiline	fluphenazine	pazopanib	acetic acid	chlorpromazine	clomifene	vandetanib	chromic chloride	sorafenib	diethylstilbestrol	clotrimazole	tofacitinib	diiodohydroxyquinoline	mifepristone	dasatinib	ibrutinib	amiodarone	epirubicin	carbidopa	montelukast	nintedanib	astemizole	doxorubicin	bosutinib
KDM4E		vorinostat	carbidopa	methyldopa	dopamine	fenoldopam
SCN5A		amitriptyline	benzocaine	aprindine	ethotoin	lamotrigine	verapamil	carbamazepine	etidocaine	mepivacaine	lorcainide	disopyramide	moricizine	gabapentin	rufinamide	encainide	mexiletine	cinchocaine	ropivacaine	nefopam	phenytoin	quinidine	riluzole	flecainide	tocainide	cocaine	eslicarbazepine acetate	dextropropoxyphene	lidocaine	fosphenytoin	topiramate	mephenytoin	oxcarbazepine	procainamide	tetracaine	propafenone	amiodarone	phenazopyridine	indecainide	ranolazine	orphenadrine	bepridil	hydroquinidine
OPRK1		meperidine	raloxifene	levorphanol	alvimopan	hydromorphone	pentazocine	naloxone	nelfinavir	saquinavir	disulfiram	oxymorphone	pimozide	loperamide	ritonavir	fentanyl	flunarizine	danazol	methadone	econazole	tamoxifen	sufentanil	ethinylestradiol	nalfurafine	thioridazine	butorphanol	cefapirin	miconazole	tramadol	eluxadoline	fluphenazine	codeine	bisacodyl	buprenorphine	hydrocodone	chlorpromazine	nalmefene	morphine	naltrexone	cocaine	domperidone	diethylstilbestrol	clotrimazole	mifepristone	amiodarone	haloprogin	dezocine	ketobemidone	nalorphine	nalbuphine	oxycodone	astemizole
OPRD1		paclitaxel	sufentanil	nalfurafine	raloxifene	butorphanol	cefapirin	miconazole	tramadol	eluxadoline	levorphanol	fluphenazine	alvimopan	codeine	buprenorphine	hydromorphone	chlorpromazine	oxiconazole	pentazocine	ketoconazole	nalmefene	chlorambucil	naloxone	morphine	nelfinavir	naltrexone	saquinavir	diethylstilbestrol	clotrimazole	oxymorphone	pimozide	loperamide	amiodarone	fentanyl	flunarizine	montelukast	ketobemidone	nalorphine	nalbuphine	oxycodone	astemizole	methadone	econazole	tamoxifen
SLC22A1		amitriptyline	irinotecan	atropine	imipramine	memantine	verapamil	metformin	clonidine	tramadol	amiloride	disopyramide	terazosin	chlorprothixene	quinine	chlorpromazine	ondansetron	flupentixol	pentamidine	trimethoprim	prazosin	apomorphine	promazine	clomipramine	amsacrine	morphine	diltiazem	mitoxantrone	prochlorperazine	repaglinide	trimipramine	desipramine	loperamide	promethazine	propafenone	propranolol	ritonavir	metoclopramide	mepenzolate	phenoxybenzamine	orphenadrine	citalopram	clemastine	nandrolone	chlorhexidine	oxprenolol	bithionol
ADRB2		pseudoephedrine	nadolol	timolol	orciprenaline	tirilazad	betaxolol	indacaterol	fenoterol	sotalol	bitolterol	xamoterol	sertindole	dopexamine	norepinephrine	penbutolol	risperidone	vortioxetine	ergotamine	tulobuterol	quetiapine	formoterol	procaterol	zotepine	bupranolol	terguride	loperamide	olanzapine	propranolol	acebutolol	alprenolol	ritodrine	dobutamine	reproterol	droxidopa	oxprenolol	fenfluramine	levobetaxolol	tretoquinol	protokylol	ziprasidone	bufuralol	terbutaline	epinephrine	levobunolol	darifenacin	salbutamol	clenbuterol	nebivolol	pipamperone	ephedrine	metoprolol	pindolol	doxazosin	celiprolol	clozapine	carteolol	bambuterol	arformoterol	dopamine	metipranolol	aripiprazole	asenapine	labetalol	bromocriptine	fluspirilene	pirbuterol	carvedilol	lisuride	levosalbutamol	olodaterol	bopindolol	haloperidol	propafenone	atenolol	montelukast	vilanterol	brexpiprazole	salmeterol	bisoprolol	paliperidone	isoprenaline	lysergic acid diethylamide
CYP51A1		fluconazole	testosterone	griseofulvin	rifampicin	tolnaftate	ketoconazole	clotrimazole	itraconazole	miconazole	terconazole	econazole	bifonazole
CYP2C9		zafirlukast	losartan	nimodipine	dicoumarol	warfarin	raloxifene	benzbromarone	candesartan cilexetil	mosapride	mefenamic acid	megestrol acetate	fluconazole	oxiconazole	idebenone	phenylbutazone	diclofenamide	felodipine	niclosamide	omeprazole	voriconazole	glyburide	propofol	tenidap	sulconazole	nitrendipine	atazanavir	ritonavir	sirolimus	danazol	suprofen	liothyronine	econazole	fluvastatin	stanozolol	pyrimethamine	ibuprofen	miconazole	noscapine	bisacodyl	nicardipine	dihydroergocristine	finasteride	lacidipine	sulfaphenazole	cilostazol	tropicamide	clotrimazole	troglitazone	gemfibrozil	amiodarone	phenelzine	mezlocillin	podofilox
HTR2B		piribedil	mitotane	cyclobenzaprine	sulfadiazine	metergoline	mosapride	ebastine	thiethylperazine	cyclizine	valdecoxib	duloxetine	prazosin	oxiconazole	apomorphine	isoflurane	propofol	risperidone	ketotifen	chloroxylenol	ergometrine	xanomeline	disulfiram	tretinoin	sulconazole	desipramine	olanzapine	alosetron	promethazine	fluoxetine	terfenadine	amisulpride	propranolol	flunarizine	orphenadrine	tamoxifen	amitriptyline	isotretinoin	ropinirole	cariprazine	trazodone	verapamil	cinnarizine	methysergide	cabergoline	dihydroergotamine	miconazole	pipamperone	chlorpromazine	clomifene	promazine	aripiprazole	clomipramine	labetalol	diphenhydramine	amoxicillin	dihydro-alpha-ergocryptine	droperidol	bromocriptine	sorafenib	lisuride	metamfetamine	buspirone	benzatropine	clotrimazole	propafenone	montelukast	oxatomide	clemastine	astemizole	guanabenz	pergolide	sertraline	dicyclomine	oxymetazoline	amoxapine	raloxifene	benzbromarone	tirilazad	flibanserin	mianserin	ondansetron	ethambutol	mexiletine	prochlorperazine	ergotamine	quetiapine	suloctidil	hexachlorophene	tegaserod	terguride	desloratadine	mepyramine	loperamide	cyproheptadine	metoclopramide	citalopram	bithionol	econazole	fenfluramine	fendiline	estradiol benzoate	nortriptyline	ziprasidone	thioridazine	cefapirin	maprotiline	ketanserin	yohimbine	agomelatine	fluphenazine	chlorpheniramine	nalidixic acid	protriptyline	pindolol	doxazosin	oxybutynin	lorcaserin	clozapine	loratadine	melatonin	asenapine	dihydroergocristine	doxepin	nefopam	aclarubicin	fluspirilene	carvedilol	domperidone	tolnaftate	pizotifen	diethylstilbestrol	methylergometrine	troglitazone	bopindolol	haloperidol	phentolamine	estrone	guanfacine	sarpogrelate	amiodarone	cisapride	dexfenfluramine	methapyrilene	brexpiprazole	dapiprazole	paliperidone	lysergic acid diethylamide
CA2		acetohydroxamic acid	mafenide	coumarin	imatinib	chlorthalidone	aminobenzoic acid	sulfanilamide	hydroxyurea	ethoxzolamide	valdecoxib	acetazolamide	hydrochlorothiazide	zonisamide	diclofenamide	cefuroxime	propofol	salicylic acid	celecoxib	pyrazinamide	sulthiame	methylparaben	bendroflumethiazide	nilotinib	triethylenetetramine	dobutamine	zoledronic acid	sulpiride	brinzolamide	cianidanol	methazolamide	chlorothiazide	trichlormethiazide	acetaminophen	pioglitazone	paraoxon	diflunisal	phenol	rosiglitazone	benzthiazide	probenecid	cinoxacin	clotrimazole	troglitazone	indapamide	tioxolone	topiramate	dorzolamide	lacosamide	ethyl hydroxybenzoate	furosemide	guaiacol	quercetin	resorcinol	sulfasalazine	mezlocillin	hydroquinone
TBXAS1		nifedipine	amprenavir	zafirlukast	trovafloxacin	imatinib	miconazole	ozagrel	candesartan cilexetil	aminoglutethimide	oxiconazole	ketoconazole	rosiglitazone	lacidipine	nelfinavir	saquinavir	ergotamine	diethylstilbestrol	hexachlorophene	clotrimazole	indinavir	troglitazone	sulconazole	ritonavir	vinblastine	montelukast	sulfasalazine	mezlocillin	bithionol	econazole	tamoxifen
MAPK1		isotretinoin	zafirlukast	sorafenib	dicoumarol	hexachlorophene	tretinoin	benzbromarone	diiodohydroxyquinoline	troglitazone	exisulind	aceclofenac	sulfasalazine	bithionol	meclofenamic acid
AKR1B1		phenylbutyric acid	tolrestat	phenylacetic acid	nitazoxanide	gossypol	troglitazone	indomethacin	sulindac	mefenamic acid	epalrestat	hymecromone	tolmetin	quercetin	flufenamic acid	mezlocillin
PTPN1		tiludronic acid	clodronic acid	quercetin	estramustine phosphate	troglitazone	aminosalicylic acid	enoxolone
AOX1		amitriptyline	nortriptyline	ethinylestradiol	perphenazine	verapamil	thioridazine	cyclobenzaprine	raloxifene	maprotiline	quinacrine	chlorpromazine	ondansetron	clozapine	ketoconazole	promazine	clomipramine	felodipine	tacrine	hydralazine	domperidone	amlodipine	quetiapine	loperamide	olanzapine	promethazine	propafenone	metoclopramide	erythromycin	salmeterol	estradiol	tamoxifen
KCNH2		nifedipine	levacetylmethadol	epinastine	telithromycin	dofetilide	phenylpropanolamine	amifampridine	mosapride	ebastine	guanidine	dolasetron	pentobarbital	prazosin	ketoconazole	donepezil	sertindole	ifenprodil	fexofenadine	arsenic trioxide	glyburide	ibutilide	risperidone	flecainide	desipramine	olanzapine	alosetron	fluoxetine	primaquine	terfenadine	caffeine	procainamide	flunarizine	orphenadrine	levofloxacin	moclobemide	bepridil	hydroquinidine	tamoxifen	amitriptyline	brompheniramine	sunitinib	beclabuvir	rimonabant	imipramine	trazodone	verapamil	granisetron	daclatasvir	mizolastine	azithromycin	miconazole	perhexiline	nisoldipine	paroxetine	quinine	chlorpromazine	clomifene	mesoridazine	aripiprazole	diphenhydramine	benperidol	quinidine	droperidol	buspirone	cibenzoline	clotrimazole	papaverine	azimilide	propafenone	cetirizine	halofantrine	ranolazine	clemastine	febuxostat	astemizole	pergolide	sertraline	dicyclomine	ouabain	meperidine	perphenazine	vesnarinone	tacrolimus	ceritinib	sildenafil	disopyramide	lumefantrine	terazosin	digoxin	ondansetron	dronedarone	sotalol	methadyl acetate	mexiletine	amsacrine	flavoxate	mitoxantrone	prochlorperazine	azelastine	bupivacaine	quetiapine	budipine	isradipine	pimozide	mepyramine	chloroquine	nitrendipine	cyproheptadine	clebopride	fentanyl	pilsicainide	citalopram	methadone	tadalafil	aprindine	ziprasidone	grepafloxacin	thioridazine	lopinavir	clarithromycin	ketanserin	fluphenazine	amodiaquine	probucol	chlorpheniramine	protriptyline	buprenorphine	tolterodine	doxazosin	pentamidine	lidoflazine	sparfloxacin	clozapine	loratadine	mefloquine	melperone	diltiazem	fasudil	fluspirilene	carvedilol	cocaine	digitoxin	domperidone	trifluoperazine	atomoxetine	haloperidol	phentolamine	mibefradil	levobupivacaine	amiodarone	osimertinib	cisapride	erythromycin	hydroxychloroquine	terodiline	dalfampridine	paliperidone
ADORA2B		caffeine	theophylline	acefylline	pentoxifylline	enprofylline	adenosine
ADORA1		nifedipine	theophylline	tinoridine	diethylstilbestrol	clotrimazole	miconazole	sildenafil	adenosine	caffeine	gabapentin	regadenoson	istradefylline	lovastatin	enprofylline	liothyronine	mefloquine	econazole	tamoxifen
PIK3CD		sunitinib	dasatinib	caffeine	idelalisib	theophylline
ACHE		irinotecan	ranitidine	edrophonium	raloxifene	physostigmine	terconazole	echothiophate	metergoline	ebastine	isoflurophate	oxiconazole	donepezil	fenofibrate	minaprine	methoxsalen	ethylestrenol	ambenonium	nizatidine	hexachlorophene	bromopride	obidoxime	fluoxetine	caffeine	procainamide	clebopride	neostigmine	econazole	rimonabant	decamethonium	miconazole	quinacrine	bambuterol	tacrine	rivastigmine	gallamine	rutin	diethylstilbestrol	profenamine	clotrimazole	galantamine	acotiamide	butenafine	papaverine	distigmine	pentoxifylline	propentofylline	ipidacrine	quercetin	pyridostigmine
ADORA2A		nifedipine	ethinylestradiol	theophylline	trioxsalen	diethylstilbestrol	hexachlorophene	raloxifene	clotrimazole	miconazole	sildenafil	amiloride	adenosine	nisoldipine	caffeine	imiquimod	regadenoson	istradefylline	enprofylline	mefloquine	bithionol	econazole	tamoxifen
PDE5A		tadalafil	dipyridamole	udenafil	mirodenafil	pentoxifylline	avanafil	sildenafil	milrinone	papaverine	vardenafil
PDE4A		nifedipine	flavoxate	losartan	chlortetracycline	cladribine	nimesulide	theophylline	roflumilast	celecoxib	amrinone	apremilast	disulfiram	ibudilast	benzbromarone	sildenafil	crisaborole	papaverine	dipyridamole	amlexanox	enoximone	milrinone	vardenafil
PDE4B		dyphylline	flavoxate	losartan	roflumilast	amrinone	ibudilast	sildenafil	crisaborole	papaverine	drotaverine	pentoxifylline	amlexanox	enoximone	enprofylline	milrinone	vardenafil
PDE4C		flavoxate	losartan	roflumilast	amrinone	amlexanox	apremilast	enoximone	ibudilast	sildenafil	crisaborole	milrinone	vardenafil
PDE4D		flavoxate	losartan	roflumilast	amrinone	amlexanox	apremilast	enoximone	ibudilast	sildenafil	crisaborole	milrinone	vardenafil
ABCC5		tioguanine	mercaptopurine	fluorouracil	methotrexate	sildenafil	azathioprine
PDE1A		dipyridamole	vinpocetine	sildenafil	crisaborole	papaverine	vardenafil
PDE3A		dyphylline	losartan	pimobendan	theophylline	vesnarinone	amrinone	cilostazol	levosimendan	sildenafil	papaverine	dipyridamole	anagrelide	enoximone	milrinone	vardenafil
PDE3B		dipyridamole	losartan	pimobendan	vesnarinone	amrinone	cilostazol	sildenafil	milrinone	papaverine	vardenafil
PDE11A		tadalafil	dipyridamole	mezlocillin	sildenafil	oxacillin	vardenafil
PDE10A		dipyridamole	cinchophen	oxycinchophen	sildenafil	papaverine	vardenafil
PDE2A		dipyridamole	dicloxacillin	anagrelide	sildenafil	papaverine	vardenafil
KCNH1		haloperidol	terfenadine	guanidine	quinidine	imipramine	dofetilide	astemizole	dalfampridine	amifampridine
KCNK2		isoflurane	enflurane	desflurane	amlodipine	sevoflurane	dofetilide	halothane
DHFR		pemetrexed	trimethoprim	aminopterin	pyrimethamine	raltitrexed	methotrexate	pralatrexate	sulfacetamide	cycloguanil	iclaprim	leucovorin	trimetrexate
SLC47A1		irinotecan	ranitidine	gabexate	telmisartan	zafirlukast	ethinylestradiol	granisetron	imatinib	pyrimethamine	clonidine	epinastine	dihydroergotamine	noscapine	amantadine	camostat	cortisone acetate	ondansetron	pentamidine	cimetidine	prazosin	rimantadine	sumatriptan	maraviroc	famotidine	dabigatran etexilate	mitoxantrone	quinidine	risperidone	carvedilol	domperidone	buspirone	indinavir	spironolactone	pantoprazole	ritonavir	levofloxacin	astemizole	chlorhexidine	bithionol	topotecan
SLC18A2		benzphetamine	valbenazine	deutetrabenazine	lisdexamfetamine	tetrabenazine	deserpidine	ketanserin	reserpine	dextroamphetamine	rescinnamine
DRD3		piribedil	rotigotine	terconazole	metergoline	ebastine	thiethylperazine	cyclizine	indacaterol	loxapine	oxiconazole	apomorphine	fenofibrate	sertindole	vilazodone	risperidone	ketotifen	ergometrine	tiapride	xanomeline	disulfiram	zotepine	sulconazole	olanzapine	promethazine	fluoxetine	terfenadine	amisulpride	flunarizine	rabeprazole	sultopride	tamoxifen	amitriptyline	ropinirole	cariprazine	imipramine	trazodone	verapamil	cyamemazine	cinnarizine	methysergide	benzquinamide	cabergoline	dihydroergotamine	miconazole	trifluperidol	pipamperone	paroxetine	chlorprothixene	chlorpromazine	clomifene	dopamine	promazine	mesoridazine	aripiprazole	bromperidol	clomipramine	benperidol	droperidol	bromocriptine	lisuride	buspirone	benzatropine	clotrimazole	thiothixene	iloperidone	haloprogin	montelukast	chlorproethazine	oxatomide	amifostine	clemastine	salmeterol	astemizole	pergolide	dicyclomine	molindone	perphenazine	amoxapine	raloxifene	flibanserin	aripiprazole lauroxil	remoxipride	mianserin	pramipexole	diphenidol	tamsulosin	prochlorperazine	saquinavir	ergotamine	quetiapine	suloctidil	formoterol	pimozide	terguride	desloratadine	loperamide	cyproheptadine	metoclopramide	clebopride	danazol	dobutamine	bithionol	econazole	sulpiride	mirtazapine	nortriptyline	ziprasidone	thioridazine	cefapirin	maprotiline	reserpine	yohimbine	fluphenazine	quinacrine	oxybutynin	flupentixol	pentamidine	thioproperazine	clozapine	asenapine	dihydroergocristine	doxepin	perospirone	lacidipine	melperone	fluspirilene	carvedilol	domperidone	diethylstilbestrol	trifluoperazine	methylergometrine	haloperidol	amiodarone	cisapride	brexpiprazole	moperone	paliperidone	lysergic acid diethylamide
DRD2		piribedil	rotigotine	tetrabenazine	metergoline	ebastine	thiethylperazine	indacaterol	loxapine	apomorphine	sertindole	vilazodone	clothiapine	gepirone	risperidone	ergometrine	tiapride	xanomeline	disulfiram	etoperidone	bromopride	zotepine	desipramine	olanzapine	promethazine	terfenadine	amisulpride	flunarizine	sultopride	triflupromazine	tamoxifen	amitriptyline	ropinirole	cariprazine	phenyltoloxamine	carphenazine	imipramine	trazodone	cyamemazine	modafinil	cinnarizine	methysergide	benzquinamide	cabergoline	dihydroergotamine	miconazole	darifenacin	trifluperidol	pipamperone	chlorprothixene	chlorpromazine	armodafinil	dopamine	promazine	mesoridazine	aripiprazole	bromperidol	clomipramine	benperidol	droperidol	bromocriptine	lisuride	buspirone	clotrimazole	thiothixene	acetophenazine	iloperidone	nefazodone	chlorproethazine	cefixime	clemastine	astemizole	pergolide	molindone	perphenazine	tandospirone	amoxapine	raloxifene	flibanserin	aripiprazole lauroxil	remoxipride	mianserin	lurasidone	pramipexole	diphenidol	tamsulosin	zuclopenthixol	prochlorperazine	blonanserin	ergotamine	quetiapine	pimozide	terguride	cyproheptadine	metoclopramide	clebopride	levodopa	econazole	sulpiride	mirtazapine	nortriptyline	ziprasidone	thioridazine	cefapirin	maprotiline	ketanserin	reserpine	alizapride	yohimbine	fluphenazine	flupentixol	thioproperazine	zimelidine	clozapine	asenapine	dihydroergocristine	doxepin	perospirone	melperone	fluspirilene	carvedilol	domperidone	pizotifen	diethylstilbestrol	trifluoperazine	methylergometrine	haloperidol	amiodarone	lofepramine	propiomazine	cisapride	brexpiprazole	fenoldopam	moperone	paliperidone	lysergic acid diethylamide
HTR1A		piribedil	clonidine	nomifensine	metergoline	ebastine	thiethylperazine	duloxetine	loxapine	oxiconazole	apomorphine	sertindole	tranylcypromine	vilazodone	brimonidine	gepirone	penbutolol	risperidone	ketotifen	ergometrine	xanomeline	etoperidone	zotepine	desipramine	olanzapine	promethazine	propranolol	flunarizine	moclobemide	tamoxifen	amitriptyline	ropinirole	cariprazine	imipramine	trazodone	verapamil	cyamemazine	cinnarizine	methysergide	cabergoline	dihydroergotamine	miconazole	zolmitriptan	pipamperone	moxonidine	paroxetine	phendimetrazine	chlorpromazine	dopamine	promazine	mesoridazine	aripiprazole	labetalol	droperidol	bromocriptine	sorafenib	lisuride	buspirone	clotrimazole	thiothixene	iloperidone	propafenone	nefazodone	urapidil	astemizole	guanabenz	pergolide	lofexidine	molindone	frovatriptan	timolol	tertatolol	perphenazine	oxymetazoline	tandospirone	amoxapine	flibanserin	aripiprazole lauroxil	remoxipride	mianserin	lurasidone	pramipexole	eletriptan	tamsulosin	rizatriptan	naratriptan	prochlorperazine	vortioxetine	saquinavir	ergotamine	quetiapine	suloctidil	tegaserod	pimozide	terguride	dextroamphetamine	cyproheptadine	bithionol	econazole	fenfluramine	mirtazapine	nortriptyline	oxitriptan	ziprasidone	thioridazine	cefapirin	levobunolol	ketanserin	reserpine	tropisetron	yohimbine	fluphenazine	clenbuterol	nebivolol	pindolol	flupentixol	clozapine	synephrine	sumatriptan	asenapine	dihydroergocristine	doxepin	melperone	fluspirilene	carvedilol	pizotifen	trifluoperazine	methylergometrine	bopindolol	haloperidol	phentolamine	lofepramine	dexfenfluramine	brexpiprazole	dapiprazole	paliperidone	lysergic acid diethylamide
DRD1		amoxapine	rotigotine	raloxifene	terconazole	metergoline	mianserin	ebastine	thiethylperazine	loxapine	oxiconazole	apomorphine	sertindole	dopexamine	zuclopenthixol	nelfinavir	prochlorperazine	risperidone	ketotifen	celecoxib	ergometrine	ergotamine	disulfiram	quetiapine	zotepine	terguride	desipramine	olanzapine	promethazine	terfenadine	cyproheptadine	flunarizine	levodopa	danazol	econazole	tamoxifen	amitriptyline	mirtazapine	nortriptyline	ropinirole	cariprazine	phenyltoloxamine	ziprasidone	trazodone	cyamemazine	methysergide	thioridazine	cabergoline	dihydroergotamine	epinephrine	maprotiline	miconazole	ketanserin	reserpine	fluphenazine	chlorprothixene	chlorpromazine	flupentixol	clozapine	dopamine	promazine	mesoridazine	aripiprazole	asenapine	bromperidol	clomipramine	dihydroergocristine	doxepin	droperidol	bromocriptine	carvedilol	lisuride	diethylstilbestrol	clotrimazole	thiothixene	methylergometrine	haloperidol	iloperidone	amiodarone	haloprogin	propiomazine	cisapride	brexpiprazole	clemastine	astemizole	fenoldopam	pergolide	paliperidone
SCN1A		dicyclomine	nifedipine	ethotoin	tetrabenazine	quinisocaine	levorphanol	mepivacaine	mianserin	hexylcaine	prilocaine	propoxycaine	prazosin	zonisamide	diphenidol	levetiracetam	mexiletine	cinchocaine	felodipine	hexobendine	ropivacaine	phenytoin	proparacaine	bupivacaine	tocainide	desipramine	pheniramine	loperamide	nitrendipine	promethazine	procainamide	cyproheptadine	flunarizine	phenoxybenzamine	orphenadrine	bepridil	prenylamine	benzocaine	brompheniramine	lamotrigine	oxetacaine	imipramine	verapamil	cinnarizine	thioridazine	reserpine	yohimbine	fluphenazine	nisoldipine	chlorpheniramine	quinacrine	quinine	chlorpromazine	rufinamide	promazine	diphenhydramine	diltiazem	quinidine	droperidol	cocaine	eslicarbazepine acetate	trifluoperazine	phenacemide	articaine	haloperidol	phentolamine	topiramate	dilazep	mephenytoin	oxybuprocaine	tetracaine	levobupivacaine	gallopamil	phenazopyridine	pramocaine
SCN2A		dicyclomine	nifedipine	ethotoin	tetrabenazine	quinisocaine	etidocaine	levorphanol	mepivacaine	mianserin	hexylcaine	prilocaine	propoxycaine	prazosin	diphenidol	mexiletine	cinchocaine	felodipine	hexobendine	ropivacaine	phenytoin	proparacaine	tocainide	lidocaine	desipramine	pheniramine	loperamide	nitrendipine	promethazine	procainamide	cyproheptadine	phenoxybenzamine	bepridil	prenylamine	amitriptyline	benzocaine	brompheniramine	lamotrigine	oxetacaine	imipramine	verapamil	cinnarizine	thioridazine	reserpine	yohimbine	fluphenazine	nisoldipine	chlorpheniramine	quinacrine	quinine	chlorpromazine	rufinamide	promazine	diphenhydramine	diltiazem	quinidine	droperidol	cocaine	eslicarbazepine acetate	trifluoperazine	articaine	haloperidol	phentolamine	dilazep	mephenytoin	oxybuprocaine	tetracaine	gallopamil	phenazopyridine	pramocaine
SCN3A		dicyclomine	nifedipine	ethotoin	tetrabenazine	quinisocaine	levorphanol	mepivacaine	mianserin	hexylcaine	prilocaine	propoxycaine	prazosin	diphenidol	cinchocaine	felodipine	hexobendine	ropivacaine	phenytoin	proparacaine	tocainide	lidocaine	desipramine	pheniramine	loperamide	nitrendipine	promethazine	procainamide	cyproheptadine	phenoxybenzamine	bepridil	prenylamine	benzocaine	brompheniramine	lamotrigine	oxetacaine	imipramine	verapamil	cinnarizine	thioridazine	reserpine	yohimbine	fluphenazine	nisoldipine	chlorpheniramine	quinacrine	quinine	chlorpromazine	rufinamide	promazine	diphenhydramine	diltiazem	quinidine	droperidol	cocaine	eslicarbazepine acetate	trifluoperazine	articaine	haloperidol	phentolamine	dilazep	mephenytoin	oxybuprocaine	tetracaine	gallopamil	phenazopyridine	pramocaine
P2RY12		prasugrel	ticagrelor	clopidogrel	epoprostenol	ticlopidine	cangrelor
ADRA2B		methylphenidate	piribedil	clonidine	phenylpropanolamine	terconazole	metergoline	mosapride	ebastine	sibutramine	loxapine	prazosin	oxiconazole	ketoconazole	apomorphine	dosulepin	sertindole	vilazodone	brimonidine	naphazoline	tramazoline	tizanidine	norepinephrine	risperidone	ketotifen	celecoxib	ergometrine	disulfiram	zotepine	sulconazole	desipramine	olanzapine	promethazine	fluoxetine	dipivefrin	rilmenidine	flunarizine	orphenadrine	rabeprazole	tamoxifen	amitriptyline	isotretinoin	ropinirole	imipramine	trazodone	cinnarizine	methysergide	benzquinamide	cabergoline	dihydroergotamine	miconazole	pipamperone	tolazoline	chlorpromazine	clomifene	xylometazoline	tolperisone	promazine	eperisone	aripiprazole	clomipramine	droperidol	bromocriptine	bunazosin	lisuride	metamfetamine	benzatropine	clotrimazole	medetomidine	thiothixene	iloperidone	guanethidine	haloprogin	nefazodone	phenylephrine	clemastine	ticlopidine	astemizole	guanabenz	pergolide	sertraline	lofexidine	molindone	perphenazine	oxymetazoline	amoxapine	raloxifene	candesartan cilexetil	mianserin	selegiline	terazosin	pramipexole	dexmedetomidine	prochlorperazine	ergotamine	quetiapine	pimozide	terguride	desloratadine	dexniguldipine	cyproheptadine	danazol	phenoxybenzamine	dobutamine	droxidopa	bithionol	econazole	fenfluramine	mirtazapine	nortriptyline	tetryzoline	ziprasidone	thioridazine	epinephrine	maprotiline	ketanserin	yohimbine	fluphenazine	quinacrine	indoramin	clozapine	asenapine	dihydroergocristine	doxepin	apraclonidine	levonordefrin	fluspirilene	carvedilol	domperidone	diethylstilbestrol	trifluoperazine	methylergometrine	mifepristone	haloperidol	phentolamine	guanfacine	amiodarone	cisapride	dexfenfluramine	methapyrilene	brexpiprazole	dexchlorpheniramine	dapiprazole	paliperidone
ADRA2C		methylphenidate	piribedil	clonidine	phenylpropanolamine	tetrabenazine	terconazole	metergoline	ebastine	sibutramine	loxapine	prazosin	oxiconazole	apomorphine	sertindole	vilazodone	brimonidine	naphazoline	tramazoline	tizanidine	norepinephrine	risperidone	zotepine	sulconazole	olanzapine	promethazine	terfenadine	amisulpride	dipivefrin	rilmenidine	flunarizine	amitriptyline	ropinirole	trazodone	cinnarizine	methysergide	benzquinamide	cabergoline	dihydroergotamine	buflomedil	pipamperone	moxonidine	tolazoline	chlorpromazine	clomifene	xylometazoline	promazine	aripiprazole	clomipramine	droperidol	bromocriptine	lisuride	metamfetamine	amlodipine	benzatropine	medetomidine	thiothixene	iloperidone	guanethidine	haloprogin	montelukast	phenylephrine	clemastine	ticlopidine	astemizole	guanabenz	pergolide	sertraline	lofexidine	irinotecan	molindone	perphenazine	oxymetazoline	amoxapine	raloxifene	tirilazad	mianserin	terazosin	lurasidone	pramipexole	tamsulosin	dexmedetomidine	prochlorperazine	ergotamine	quetiapine	suloctidil	hexachlorophene	pimozide	terguride	dexniguldipine	cyproheptadine	danazol	droxidopa	bithionol	fenfluramine	estradiol benzoate	mirtazapine	nortriptyline	tetryzoline	ziprasidone	thioridazine	cefapirin	epinephrine	maprotiline	alizapride	yohimbine	fluphenazine	quinacrine	indoramin	emetine	doxazosin	clozapine	asenapine	dihydroergocristine	doxepin	apraclonidine	levonordefrin	fluspirilene	carvedilol	domperidone	rutin	diethylstilbestrol	trifluoperazine	haloperidol	phentolamine	guanfacine	cisapride	dexfenfluramine	brexpiprazole	paliperidone
CYP2D6		oxymetazoline	amoxapine	physostigmine	dextromethorphan	lansoprazole	metergoline	cyclizine	oxiconazole	diphenidol	doxapram	bupropion	idebenone	naloxone	amsacrine	ajmaline	rizatriptan	prochlorperazine	risperidone	bupivacaine	celecoxib	trihexyphenidyl	hydroxyzine	sulconazole	ambroxol	mepyramine	loperamide	promethazine	fluoxetine	propranolol	ritonavir	metoclopramide	orphenadrine	econazole	aprindine	nortriptyline	bufuralol	terbinafine	stanozolol	thioridazine	cefapirin	miconazole	bromhexine	perhexiline	yohimbine	diphenylpyraline	chlorpheniramine	paroxetine	chlorpromazine	clomifene	bambuterol	promazine	eperisone	clomipramine	labetalol	diphenhydramine	carmofur	melperone	tacrine	quinidine	naltrexone	valethamate	domperidone	lisuride	triamterene	atomoxetine	butenafine	methylergometrine	bopindolol	phentolamine	levobupivacaine	propafenone	cisapride	methapyrilene	clemastine	phenelzine	ticlopidine	pergolide
PTGS2		diclofenac	dexamethasone	dexibuprofen	isoxicam	oxaprozin	acetylsalicylic acid	mefenamic acid	fenbufen	tolfenamic acid	valdecoxib	monobenzone	isoflurophate	meclofenamic acid	oxacillin	tiaprofenic acid	balsalazide	mesalazine	nimesulide	celecoxib	parecoxib	hexachlorophene	tenidap	piroxicam	proquazone	ketorolac	nitroxoline	etoricoxib	thalidomide	tolmetin	loxoprofen	suprofen	bromfenac	flufenamic acid	tamoxifen	nabumetone	flurbiprofen	cianidanol	cefonicid	benzquinamide	ibuprofen	alclofenac	miconazole	indobufen	acemetacin	aminosalicylic acid	lumiracoxib	fenoprofen	rofecoxib	acetaminophen	ketoprofen	pirprofen	dexketoprofen	niflumic acid	captopril	zomepirac	aceclofenac	tenoxicam	diflunisal	carprofen	cefotetan	nepafenac	bismuth subsalicylate	oxyphenbutazone	etodolac	clotrimazole	cefalotin	indomethacin	sulindac	naproxen	meloxicam	felbinac	quercetin	sulfasalazine	ticlopidine	mezlocillin	aminophenazone	floctafenine
RARA		isotretinoin	acitretin	bexarotene	tazarotene	adapalene	alitretinoin	tretinoin	tamibarotene	etretinate
RARG		acitretin	bexarotene	tazarotene	adapalene	alitretinoin	rosiglitazone	tretinoin	tamibarotene
RARB		isotretinoin	bexarotene	tazarotene	adapalene	alitretinoin	tretinoin	tamibarotene
HSP90AA1		famotidine	primaquine	terfenadine	midodrine	formoterol
SLC22A2		amitriptyline	irinotecan	gabexate	zafirlukast	ethinylestradiol	imipramine	verapamil	granisetron	imatinib	metformin	clonidine	epinastine	dihydroergotamine	noscapine	camostat	sibutramine	chlorpromazine	ondansetron	pentamidine	prazosin	rimantadine	mexiletine	diphenhydramine	doxepin	famotidine	dabigatran etexilate	mitoxantrone	quinidine	risperidone	carvedilol	domperidone	buspirone	flurazepam	ipratropium	pimozide	pantoprazole	propafenone	ritonavir	chlorhexidine	bithionol	topotecan	tamoxifen
SLC47A2		famotidine	irinotecan	gabexate	dabigatran etexilate	zafirlukast	mitoxantrone	ethinylestradiol	domperidone	buspirone	imatinib	epinastine	dihydroergotamine	indinavir	camostat	pantoprazole	ritonavir	ondansetron	pentamidine	cimetidine	prazosin	chlorhexidine	bithionol	topotecan
ATP4A		omeprazole	pantoprazole	dexrabeprazole	dexlansoprazole	esomeprazole	ilaprazole	lansoprazole	rabeprazole	vonoprazan
ATP4B		omeprazole	pantoprazole	dexrabeprazole	dexlansoprazole	esomeprazole	ilaprazole	lansoprazole	rabeprazole	vonoprazan
ATP1A1		deslanoside	metildigoxin	ouabain	pantoprazole	digoxin	bumetanide	digitoxin	proscillaridin	furosemide	rabeprazole	acetyldigitoxin
FASN		omeprazole	pantoprazole	cerulenin	lansoprazole	rabeprazole
SLC12A1		etacrynic acid	bumetanide	triamterene	furosemide	torasemide	metolazone	piretanide
ADRA1D		piribedil	terconazole	metergoline	nylidrin	ebastine	cyclizine	prazosin	ketoconazole	apomorphine	vilazodone	brimonidine	norepinephrine	risperidone	ketotifen	olanzapine	promethazine	terfenadine	flunarizine	tamoxifen	amitriptyline	atropine	cariprazine	trazodone	verapamil	cinnarizine	cabergoline	dihydroergotamine	miconazole	buflomedil	chlorpromazine	promazine	clomipramine	labetalol	tacrine	droperidol	bromocriptine	lisuride	buspirone	amlodipine	benzatropine	clotrimazole	medetomidine	propafenone	guanethidine	phenylephrine	urapidil	clemastine	astemizole	guanabenz	pergolide	methoxamine	oxymetazoline	amoxapine	raloxifene	silodosin	mianserin	alfuzosin	terazosin	imiquimod	tamsulosin	dexmedetomidine	prochlorperazine	ergotamine	quetiapine	terguride	loperamide	dexniguldipine	naftopidil	cyproheptadine	dobutamine	citalopram	droxidopa	econazole	nortriptyline	tetryzoline	thioridazine	epinephrine	maprotiline	ketanserin	yohimbine	fluphenazine	quinacrine	indoramin	emetine	doxazosin	pentamidine	clozapine	dihydroergocristine	doxepin	apraclonidine	levonordefrin	carvedilol	domperidone	diethylstilbestrol	haloperidol	phentolamine	guanfacine	cisapride	hydroxychloroquine	brexpiprazole	fenoldopam	dexchlorpheniramine	dapiprazole
HTR2C		nifedipine	cyclobenzaprine	terconazole	metergoline	mosapride	ebastine	thiethylperazine	cyclizine	duloxetine	loxapine	apomorphine	fenofibrate	sertindole	propofol	risperidone	ketotifen	ergometrine	xanomeline	zotepine	sulconazole	desipramine	olanzapine	promethazine	fluoxetine	terfenadine	propranolol	flunarizine	orphenadrine	escitalopram	tamoxifen	amitriptyline	atropine	cariprazine	imipramine	trazodone	verapamil	cyamemazine	methysergide	cabergoline	dihydroergotamine	miconazole	pipamperone	chlorpromazine	clomifene	pimavanserin	promazine	mesoridazine	aripiprazole	clomipramine	diphenhydramine	amoxicillin	droperidol	bromocriptine	sorafenib	lisuride	buspirone	benzatropine	clotrimazole	thiothixene	tetracaine	iloperidone	propafenone	haloprogin	nefazodone	clemastine	astemizole	guanabenz	pergolide	reboxetine	sertraline	dicyclomine	molindone	perphenazine	oxymetazoline	raloxifene	tirilazad	flibanserin	aripiprazole lauroxil	mianserin	ethambutol	rizatriptan	mitoxantrone	prochlorperazine	vortioxetine	ergotamine	quetiapine	hexachlorophene	pimozide	terguride	desloratadine	mepyramine	venlafaxine	cyproheptadine	penfluridol	metoclopramide	metixene	citalopram	bithionol	econazole	fenfluramine	mirtazapine	nortriptyline	ziprasidone	thioridazine	maprotiline	ketanserin	agomelatine	fluphenazine	protriptyline	pindolol	doxazosin	lorcaserin	pentamidine	clozapine	sumatriptan	asenapine	dihydroergocristine	doxepin	melperone	nefopam	trioxsalen	carvedilol	domperidone	pizotifen	diethylstilbestrol	trifluoperazine	methylergometrine	haloperidol	phentolamine	guanfacine	sarpogrelate	amiodarone	lofepramine	propiomazine	cisapride	dexfenfluramine	methapyrilene	brexpiprazole	dexchlorpheniramine	dapiprazole	paliperidone	lysergic acid diethylamide
HRH1		epinastine	cyclobenzaprine	nomifensine	carbamazepine	metergoline	ebastine	carbinoxamine	thiethylperazine	cyclizine	duloxetine	loxapine	talastine	dosulepin	sertindole	ifenprodil	vilazodone	fexofenadine	risperidone	ketotifen	acrivastine	etoperidone	zotepine	chlordiazepoxide	desipramine	pheniramine	olanzapine	levocetirizine	promethazine	fluoxetine	terfenadine	mazindol	propranolol	flunarizine	orphenadrine	escitalopram	methdilazine	bilastine	amitriptyline	brompheniramine	atropine	cariprazine	phenyltoloxamine	bamipine	imipramine	trazodone	cinnarizine	methysergide	mizolastine	rupatadine	pipamperone	chlorprothixene	chlorpromazine	clomifene	antazoline	promazine	mesoridazine	aripiprazole	bromperidol	clomipramine	diphenhydramine	histamine	olopatadine	droperidol	aceprometazine	lisuride	benzatropine	clotrimazole	thiothixene	iloperidone	cetirizine	nefazodone	iprindole	oxatomide	triprolidine	clemastine	astemizole	mebhydrolin	molindone	meclizine	perphenazine	tripelennamine	amoxapine	aripiprazole lauroxil	mianserin	disopyramide	bepotastine	bromodiphenhydramine	dexbrompheniramine	dimetindene	methotrimeprazine	azatadine	doxylamine	prochlorperazine	azelastine	alcaftadine	vortioxetine	quetiapine	suloctidil	hydroxyzine	pimozide	desloratadine	mepyramine	loperamide	pitolisant	cyproheptadine	emedastine	citalopram	mirtazapine	nortriptyline	buclizine	ziprasidone	thioridazine	maprotiline	ketanserin	fluphenazine	diphenylpyraline	chlorpheniramine	protriptyline	levocabastine	flupentixol	clozapine	loratadine	asenapine	doxepin	melperone	fluspirilene	cocaine	domperidone	trifluoperazine	trimipramine	haloperidol	phentolamine	alimemazine	lofepramine	propiomazine	mequitazine	methapyrilene	brexpiprazole	dexchlorpheniramine	paliperidone	lysergic acid diethylamide
HTR2A		nifedipine	zidovudine	epinastine	cyclobenzaprine	sulfadiazine	terconazole	metergoline	ebastine	thiethylperazine	cyclizine	cimetidine	duloxetine	loxapine	prazosin	oxiconazole	apomorphine	fenofibrate	dosulepin	sertindole	risperidone	ketotifen	ergometrine	xanomeline	zotepine	sulconazole	desipramine	olanzapine	promethazine	fluoxetine	terfenadine	amisulpride	propranolol	flunarizine	alprenolol	orphenadrine	triflupromazine	tamoxifen	amitriptyline	atropine	cariprazine	carphenazine	imipramine	trazodone	verapamil	cyamemazine	cinnarizine	methysergide	cabergoline	dihydroergotamine	miconazole	pipamperone	chlorprothixene	chlorpromazine	clomifene	pimavanserin	promazine	mesoridazine	aripiprazole	clomipramine	diphenhydramine	amoxicillin	benperidol	droperidol	bromocriptine	sorafenib	lisuride	buspirone	benzatropine	clotrimazole	thiothixene	naftidrofuryl	tetracaine	iloperidone	propafenone	haloprogin	nefazodone	oxatomide	clemastine	astemizole	guanabenz	pergolide	sertraline	dicyclomine	flucytosine	molindone	perphenazine	imatinib	oxymetazoline	amoxapine	raloxifene	tirilazad	flibanserin	aripiprazole lauroxil	remoxipride	mianserin	terazosin	ethambutol	lurasidone	diphenidol	rizatriptan	zuclopenthixol	prochlorperazine	blonanserin	vortioxetine	ergotamine	quetiapine	pimozide	terguride	desloratadine	mepyramine	venlafaxine	cyproheptadine	metoclopramide	danazol	citalopram	econazole	fenfluramine	mirtazapine	nortriptyline	oxitriptan	ziprasidone	thioridazine	maprotiline	ketanserin	agomelatine	fluphenazine	protriptyline	quinacrine	pindolol	flupentixol	lorcaserin	pentamidine	clozapine	sumatriptan	asenapine	dihydroergocristine	doxepin	melperone	diltiazem	nefopam	fluspirilene	carvedilol	domperidone	pizotifen	diethylstilbestrol	trifluoperazine	methylergometrine	bopindolol	haloperidol	phentolamine	guanfacine	sarpogrelate	amiodarone	propiomazine	cisapride	dexfenfluramine	methapyrilene	brexpiprazole	dexchlorpheniramine	dapiprazole	paliperidone	lysergic acid diethylamide
HTR1F		rizatriptan	naratriptan	risperidone	xanomeline	ergotamine	methysergide	quetiapine	dihydroergotamine	zolmitriptan	ketanserin	methylergometrine	almotriptan	yohimbine	metergoline	mianserin	haloperidol	olanzapine	pipamperone	clozapine	duloxetine	eletriptan	sertindole	sumatriptan
HTR1E		ziprasidone	methysergide	oxymetazoline	thioridazine	dihydroergotamine	zolmitriptan	yohimbine	fluphenazine	metergoline	pipamperone	chlorpromazine	clozapine	duloxetine	loxapine	eletriptan	sertindole	sumatriptan	aripiprazole	asenapine	rizatriptan	naratriptan	risperidone	fluspirilene	ergometrine	xanomeline	ergotamine	quetiapine	zotepine	methylergometrine	haloperidol	olanzapine	paliperidone	lysergic acid diethylamide
HTR1B		frovatriptan	oxymetazoline	almotriptan	aripiprazole lauroxil	metergoline	mianserin	duloxetine	loxapine	pramipexole	apomorphine	eletriptan	sertindole	rizatriptan	naratriptan	risperidone	vortioxetine	xanomeline	ergotamine	quetiapine	zotepine	terguride	desipramine	olanzapine	amisulpride	propranolol	fenfluramine	ziprasidone	methysergide	thioridazine	cabergoline	dihydroergotamine	zolmitriptan	ketanserin	yohimbine	fluphenazine	pipamperone	pindolol	chlorpromazine	xylometazoline	clozapine	sumatriptan	aripiprazole	asenapine	bromocriptine	fluspirilene	cocaine	lisuride	thiothixene	haloperidol	iloperidone	dexfenfluramine	brexpiprazole	pergolide	paliperidone
HTR1D		frovatriptan	oxymetazoline	raloxifene	almotriptan	aripiprazole lauroxil	metergoline	mianserin	duloxetine	loxapine	prazosin	pramipexole	apomorphine	eletriptan	sertindole	rizatriptan	naratriptan	risperidone	vortioxetine	ergometrine	xanomeline	ergotamine	quetiapine	tegaserod	zotepine	pimozide	terguride	olanzapine	amisulpride	cyproheptadine	propranolol	rabeprazole	fenfluramine	ropinirole	ziprasidone	trazodone	methysergide	thioridazine	cabergoline	dihydroergotamine	zolmitriptan	ketanserin	yohimbine	fluphenazine	pipamperone	pindolol	chlorpromazine	xylometazoline	clozapine	sumatriptan	aripiprazole	asenapine	dihydroergocristine	melperone	bromocriptine	fluspirilene	lisuride	thiothixene	haloperidol	iloperidone	dexfenfluramine	pergolide	paliperidone	lysergic acid diethylamide
ADRB3		tretoquinol	nadolol	timolol	tertatolol	miconazole	levobunolol	candesartan cilexetil	fluphenazine	ebastine	pindolol	clomifene	oxiconazole	fenofibrate	xamoterol	arformoterol	dihydroergocristine	nelfinavir	norepinephrine	mirabegron	carvedilol	celecoxib	suloctidil	formoterol	clotrimazole	bupranolol	olodaterol	bopindolol	propafenone	propranolol	amiodarone	alprenolol	danazol	montelukast	ritodrine	vilanterol	salmeterol	astemizole	droxidopa	bisoprolol	econazole	isoprenaline	tamoxifen
EGFR		axitinib	olmutinib	sunitinib	zafirlukast	erlotinib	imatinib	thioridazine	methyldopa	gefitinib	miconazole	tirilazad	ceritinib	candesartan cilexetil	perhexiline	fluphenazine	ebastine	afatinib	crizotinib	chlorpromazine	clomifene	vandetanib	niclosamide	nelfinavir	mitoxantrone	chromic chloride	lenvatinib	ruboxistaurin	suloctidil	hexachlorophene	clotrimazole	diiodohydroxyquinoline	lapatinib	dasatinib	terfenadine	ibrutinib	docetaxel	levodopa	osimertinib	montelukast	dobutamine	quercetin	astemizole	bithionol	econazole	bosutinib	icotinib	tamoxifen
MAPK3		carmofur	nelfinavir	zafirlukast	tioguanine	hydroxyprogesterone caproate	sorafenib	disulfiram	hexachlorophene	tirilazad	diiodohydroxyquinoline
MAPK14		isotretinoin	nelfinavir	zafirlukast	sorafenib	celecoxib	imatinib	diethylstilbestrol	hexachlorophene	benzbromarone	tirilazad	diiodohydroxyquinoline	mifepristone	nilotinib	afatinib	dasatinib	etoricoxib	montelukast	fenbendazole	bithionol
ABCC9		nateglinide	glyburide	propafenone	glibornuride	pinacidil	repaglinide	gliclazide	minoxidil	glimepiride
KCNJ11		nateglinide	glyburide	acetohexamide	gliquidone	repaglinide	cibenzoline	gliclazide	levosimendan	mitiglinide	tolbutamide	glimepiride	chlorpropamide	glisoxepide	diazoxide	propafenone	glibornuride	nicorandil	carbutamide	pinacidil	glipizide	minoxidil	tolazamide
ABCC8		nateglinide	glyburide	acetohexamide	gliquidone	repaglinide	gliclazide	mitiglinide	tolbutamide	glimepiride	chlorpropamide	glisoxepide	diazoxide	glibornuride	carbutamide	glipizide	tolazamide
HCAR2		nicotinamide	acipimox	lovastatin	dimethyl fumarate	niacin
NR1I2		paclitaxel	nimodipine	raloxifene	carbamazepine	rifaximin	phenobarbital	loratadine	etoposide	nicardipine	ketoconazole	fulvestrant	rifampicin	flutrimazole	pleconaril	diethylstilbestrol	clotrimazole	isradipine	mifepristone	spironolactone	topiramate	ritonavir	bosentan	lovastatin	efavirenz	topotecan	tamoxifen
HDAC6		vorinostat	romidepsin	bufexamac	lovastatin	atorvastatin	bendamustine	panobinostat
HDAC1		phenylbutyric acid	vorinostat	romidepsin	lovastatin	valproic acid	atorvastatin	bendamustine	panobinostat
HDAC2		phenylbutyric acid	vorinostat	romidepsin	lovastatin	valproic acid	atorvastatin	bendamustine	panobinostat
KCNK10		isoflurane	enflurane	desflurane	sevoflurane	halothane
KCNK18		isoflurane	enflurane	desflurane	sevoflurane	halothane
KCNK3		isoflurane	enflurane	desflurane	sevoflurane	halothane	doxapram
KCNK9		isoflurane	enflurane	desflurane	sevoflurane	halothane	doxapram
MMP9		cefotetan	cefotiam	cefuroxime	cefonicid	flucloxacillin	secobarbital	cefalotin	aminoquinuride	budesonide	busulfan	dacarbazine	prazosin	cefradine	zoledronic acid	quercetin	beclomethasone dipropionate	chlorhexidine	econazole
NR1I3		acetaminophen	meclizine	phenobarbital	phenytoin	cerivastatin	fluvastatin	temazepam	thioridazine	simvastatin	clotrimazole	atorvastatin
GABRB2		zopiclone	prazepam	amoxapine	secobarbital	carbamazepine	eltanolone	flunitrazepam	pentobarbital	methoxyflurane	triclofos	isoflurane	propofol	triazolam	ethanol	butabarbital	chlordiazepoxide	bromazepam	nitrazepam	clonazepam	midazolam	thiopental	liothyronine	progabide	flumazenil	nordazepam	primidone	zaleplon	temazepam	fospropofol	etizolam	metharbital	estazolam	zolpidem	phenobarbital	thiamylal	delorazepam	sevoflurane	etomidate	thiocolchicoside	alfaxalone	adinazolam	alprazolam	talbutal	diazepam	eszopiclone	desflurane	flurazepam	halazepam	topiramate	clobazam	methaqualone	halothane
SLC12A3		cyclothiazide	polythiazide	chlorothiazide	chlorthalidone	trichlormethiazide	indapamide	metolazone	bendroflumethiazide	hydroflumethiazide	quinethazone	hydrochlorothiazide	methyclothiazide	benzthiazide
HTR6		amperozide	dicyclomine	molindone	perphenazine	mitotane	oxymetazoline	amoxapine	cyclobenzaprine	raloxifene	metergoline	mianserin	dapsone	ebastine	sulfadimethoxine	duloxetine	loxapine	sertindole	flutamide	zuclopenthixol	prochlorperazine	risperidone	ketotifen	vortioxetine	ergometrine	xanomeline	ergotamine	disulfiram	quetiapine	zotepine	pimozide	desloratadine	olanzapine	promethazine	terfenadine	venlafaxine	amisulpride	cyproheptadine	propranolol	orphenadrine	econazole	fenfluramine	tamoxifen	amitriptyline	nortriptyline	ziprasidone	methysergide	thioridazine	maprotiline	miconazole	ketanserin	yohimbine	fluphenazine	chlorprothixene	chlorpromazine	clomifene	clozapine	toremifene	promazine	sumatriptan	mesoridazine	aripiprazole	asenapine	clomipramine	doxepin	bromocriptine	fluspirilene	sorafenib	carvedilol	lisuride	amlodipine	diethylstilbestrol	benzatropine	clotrimazole	thiothixene	trifluoperazine	methylergometrine	haloperidol	iloperidone	propafenone	amiodarone	haloprogin	dexfenfluramine	methapyrilene	brexpiprazole	clemastine	astemizole	paliperidone	reboxetine	lysergic acid diethylamide
HRH2		dicyclomine	ranitidine	dicloxacillin	imatinib	epinastine	tirilazad	metergoline	mianserin	ebastine	imiquimod	cimetidine	loxapine	ketoconazole	pramipexole	famotidine	risperidone	ketotifen	vortioxetine	nizatidine	suloctidil	zotepine	desloratadine	loperamide	olanzapine	promethazine	cyproheptadine	orphenadrine	niperotidine	econazole	tamoxifen	amitriptyline	nortriptyline	roxatidine acetate	ziprasidone	trazodone	verapamil	thioridazine	cefapirin	maprotiline	miconazole	fluphenazine	quinacrine	chlorpromazine	clozapine	medroxyprogesterone acetate	promazine	asenapine	clomipramine	doxepin	histamine	lisuride	benzatropine	clotrimazole	thiothixene	haloperidol	amiodarone	betazole	clemastine	astemizole	dexchlorpheniramine	paliperidone
DRD4		molindone	piribedil	perphenazine	tandospirone	amoxapine	rotigotine	flibanserin	aripiprazole lauroxil	remoxipride	mianserin	ebastine	loxapine	prazosin	pramipexole	apomorphine	sertindole	prochlorperazine	risperidone	prucalopride	tiapride	disulfiram	quetiapine	zotepine	pimozide	terguride	olanzapine	amisulpride	clebopride	econazole	sulpiride	tamoxifen	ropinirole	phenyltoloxamine	ziprasidone	trazodone	thioridazine	benzquinamide	cabergoline	cefapirin	miconazole	ketanserin	trifluperidol	fluphenazine	indoramin	chlorprothixene	chlorpromazine	flupentixol	clozapine	dopamine	mesoridazine	aripiprazole	asenapine	bromperidol	benperidol	perospirone	melperone	droperidol	bromocriptine	fluspirilene	lisuride	buspirone	clotrimazole	thiothixene	trifluoperazine	haloperidol	iloperidone	amiodarone	propiomazine	chlorproethazine	brexpiprazole	quercetin	astemizole	fenoldopam	moperone	pergolide	paliperidone	lysergic acid diethylamide
HTR5A		ziprasidone	methysergide	thioridazine	dihydroergotamine	flibanserin	ketanserin	yohimbine	fluphenazine	metergoline	chlorpromazine	clozapine	loxapine	sumatriptan	aripiprazole	asenapine	risperidone	sorafenib	vortioxetine	ergotamine	quetiapine	thiothixene	zotepine	haloperidol	olanzapine	brexpiprazole	mebhydrolin	paliperidone	lysergic acid diethylamide
ADRA1B		piribedil	methoxamine	oxymetazoline	clonidine	silodosin	mianserin	nylidrin	alfuzosin	terazosin	loxapine	prazosin	apomorphine	tamsulosin	vilazodone	brimonidine	dexmedetomidine	norepinephrine	azelastine	risperidone	ergometrine	xanomeline	quetiapine	zotepine	terguride	olanzapine	dexniguldipine	terfenadine	naftopidil	cyproheptadine	droxidopa	fenfluramine	tetryzoline	ziprasidone	modafinil	thioridazine	cabergoline	dihydroergotamine	epinephrine	ketanserin	buflomedil	yohimbine	fluphenazine	indoramin	chlorpromazine	doxazosin	armodafinil	clozapine	aripiprazole	asenapine	dihydroergocristine	apraclonidine	bromocriptine	bunazosin	domperidone	lisuride	amlodipine	medetomidine	thiothixene	haloperidol	phentolamine	guanethidine	propiomazine	phenylephrine	dexfenfluramine	urapidil	brexpiprazole	fenoldopam	pergolide	dapiprazole	paliperidone
DRD5		amitriptyline	ropinirole	phenyltoloxamine	ziprasidone	thioridazine	rotigotine	cabergoline	maprotiline	ketanserin	fluphenazine	chlorprothixene	chlorpromazine	flupentixol	clozapine	loxapine	apomorphine	dopamine	aripiprazole	asenapine	risperidone	bromocriptine	lisuride	ergotamine	quetiapine	thiothixene	zotepine	terguride	haloperidol	olanzapine	iloperidone	fenoldopam	pergolide	paliperidone	lysergic acid diethylamide
HTR7		molindone	perphenazine	amoxapine	cyclobenzaprine	phenylpropanolamine	aripiprazole lauroxil	metergoline	mianserin	lurasidone	duloxetine	pramipexole	sertindole	tamsulosin	risperidone	vortioxetine	xanomeline	quetiapine	zotepine	pimozide	olanzapine	amisulpride	cyproheptadine	fenfluramine	amitriptyline	mirtazapine	ropinirole	cariprazine	oxitriptan	ziprasidone	trazodone	cyamemazine	methysergide	thioridazine	dihydroergotamine	ketanserin	yohimbine	fluphenazine	chlorpromazine	clozapine	sumatriptan	aripiprazole	asenapine	doxepin	sorafenib	pizotifen	thiothixene	trifluoperazine	haloperidol	iloperidone	cisapride	dexfenfluramine	brexpiprazole	paliperidone	lysergic acid diethylamide
G6PD		dapsone	primaquine	prasterone	nitrofural	nitrofurantoin
SLC28A1		nifedipine	dipyridamole	nimodipine	leflunomide	progesterone	sirolimus	disulfiram	diethylstilbestrol	ketoconazole	astemizole	terconazole	prednisone
SCN8A		benzocaine	ethotoin	mephenytoin	ropivacaine	phenytoin	procainamide	lamotrigine	rufinamide	tocainide	eslicarbazepine acetate	phenazopyridine	mepivacaine
SCN9A		amitriptyline	benzocaine	ethotoin	ropivacaine	phenytoin	lamotrigine	tocainide	eslicarbazepine acetate	carbamazepine	lidocaine	mepivacaine	mephenytoin	safinamide	lacosamide	procainamide	tetracaine	rufinamide	phenazopyridine	orphenadrine	mexiletine
SCN4A		benzocaine	ethotoin	ropivacaine	phenytoin	lamotrigine	bupivacaine	flecainide	tocainide	eslicarbazepine acetate	carbamazepine	etidocaine	lidocaine	mepivacaine	mephenytoin	procainamide	levobupivacaine	rufinamide	phenazopyridine	orphenadrine	pilsicainide	mexiletine
MMP2		cefotetan	cefuroxime	aclarubicin	oxyquinoline	ubenimex	doxycycline	daunorubicin	sulindac	tiludronic acid	zoledronic acid	quercetin	chlorhexidine	doxorubicin
ESR2		chlorotrianisene	ethinylestradiol	fulvestrant	diethylstilbestrol	hexachlorophene	raloxifene	estramustine phosphate	moxestrol	lasofoxifene	mifepristone	spironolactone	demeclocycline	androstenediol	estriol	estrone	bazedoxifene	ethyl hydroxybenzoate	benserazide	medroxyprogesterone acetate	bithionol	estradiol	tamoxifen
CYSLTR1		nedocromil	zafirlukast	pranlukast	montelukast	diethylstilbestrol	clotrimazole	cinalukast
PTAFR		alprazolam	brotizolam	clotrimazole	triazolam	rupatadine
TACR1		aprepitant	paroxetine	fosaprepitant	rolapitant	casopitant	cefapirin	clotrimazole	miconazole	astemizole	econazole	netupitant	tamoxifen
ERBB2		paclitaxel	erlotinib	gefitinib	miconazole	candesartan cilexetil	fluphenazine	ebastine	afatinib	chlorpromazine	clomifene	vandetanib	mitoxantrone	hexachlorophene	clotrimazole	diiodohydroxyquinoline	lapatinib	dasatinib	ibrutinib	amiodarone	astemizole	doxorubicin	bithionol	econazole	bosutinib	tamoxifen
CYP17A1		testosterone propionate	isoconazole	ketoconazole	clotrimazole	miconazole	econazole	bifonazole	tioconazole
NR1H4		felodipine	obeticholic acid	fulvestrant	nimodipine	ursodeoxycholic acid	flutrimazole	loratadine	raloxifene	clotrimazole	levothyroxine	sulconazole	chenodeoxycholic acid
MDH1		delavirdine	nicardipine	clotrimazole	miconazole	econazole	sulconazole
CCR4		amiodarone	disulfiram	quercetin	clotrimazole	itraconazole	plerixafor
KCNA3		guanidine	verapamil	diphenoxylate	clotrimazole	dalfampridine	amifampridine
CA5A		brinzolamide	mafenide	cianidanol	coumarin	methazolamide	imatinib	chlorthalidone	trichlormethiazide	sulfanilamide	hydroxyurea	ethoxzolamide	valdecoxib	acetazolamide	zonisamide	diclofenamide	celecoxib	indapamide	topiramate	nilotinib	triethylenetetramine	dorzolamide	lacosamide	dobutamine	furosemide	quercetin	resorcinol	hydroquinone	sulpiride
CA14		brinzolamide	mafenide	cianidanol	coumarin	methazolamide	imatinib	chlorthalidone	trichlormethiazide	sulfanilamide	acetaminophen	ethoxzolamide	valdecoxib	acetazolamide	zonisamide	phenol	diclofenamide	salicylic acid	celecoxib	methylparaben	indapamide	topiramate	nilotinib	triethylenetetramine	dorzolamide	lacosamide	ethyl hydroxybenzoate	dobutamine	furosemide	zoledronic acid	quercetin	resorcinol	hydroquinone
CA7		brinzolamide	mafenide	cianidanol	coumarin	methazolamide	imatinib	chlorthalidone	trichlormethiazide	sulfanilamide	acetaminophen	ethoxzolamide	valdecoxib	acetazolamide	zonisamide	diclofenamide	salicylic acid	celecoxib	methylparaben	indapamide	metolazone	topiramate	nilotinib	triethylenetetramine	dorzolamide	lacosamide	ethyl hydroxybenzoate	dobutamine	furosemide	quercetin	hesperetin	sulpiride
CA12		brinzolamide	mafenide	cianidanol	coumarin	methazolamide	imatinib	chlorthalidone	trichlormethiazide	sulfanilamide	acetaminophen	ethoxzolamide	valdecoxib	acetazolamide	zonisamide	phenol	diclofenamide	probenecid	salicylic acid	celecoxib	methylparaben	indapamide	topiramate	nilotinib	triethylenetetramine	dorzolamide	lacosamide	ethyl hydroxybenzoate	hymecromone	dobutamine	furosemide	zoledronic acid	quercetin	resorcinol	hesperetin	hydroquinone	sulpiride
CA9		brinzolamide	mafenide	cianidanol	coumarin	methazolamide	imatinib	chlorthalidone	trichlormethiazide	sulfanilamide	hydroxyurea	acetaminophen	ethoxzolamide	valdecoxib	acetazolamide	zonisamide	phenol	diclofenamide	probenecid	salicylic acid	celecoxib	sulthiame	methylparaben	indapamide	topiramate	nilotinib	triethylenetetramine	dorzolamide	lacosamide	ethyl hydroxybenzoate	hymecromone	dobutamine	furosemide	zoledronic acid	quercetin	resorcinol	hydroquinone	sulpiride
CA4		brinzolamide	mafenide	cianidanol	coumarin	methazolamide	imatinib	chlorthalidone	trichlormethiazide	sulfanilamide	acetaminophen	ethoxzolamide	valdecoxib	acetazolamide	hydrochlorothiazide	zonisamide	phenol	benzthiazide	diclofenamide	salicylic acid	celecoxib	indapamide	topiramate	bendroflumethiazide	nilotinib	triethylenetetramine	dorzolamide	lacosamide	dobutamine	furosemide	quercetin	hesperetin	hydroquinone
CA1		brinzolamide	mafenide	cianidanol	coumarin	methazolamide	verapamil	imatinib	chlorthalidone	aminobenzoic acid	trichlormethiazide	sulfanilamide	acetaminophen	paraoxon	ethoxzolamide	valdecoxib	acetazolamide	hydrochlorothiazide	zonisamide	diflunisal	phenol	levetiracetam	benzthiazide	diclofenamide	propofol	salicylic acid	celecoxib	sulthiame	amlodipine	methylparaben	indapamide	topiramate	bendroflumethiazide	nilotinib	triethylenetetramine	dorzolamide	lacosamide	ethyl hydroxybenzoate	methocarbamol	dobutamine	furosemide	guaiacol	quercetin	sulfasalazine	hydroquinone	sulpiride
CA5B		brinzolamide	mafenide	cianidanol	coumarin	methazolamide	imatinib	chlorthalidone	trichlormethiazide	sulfanilamide	ethoxzolamide	valdecoxib	acetazolamide	zonisamide	diclofenamide	celecoxib	indapamide	topiramate	nilotinib	triethylenetetramine	dorzolamide	lacosamide	dobutamine	furosemide	quercetin	resorcinol	hydroquinone	sulpiride
CA3		cianidanol	coumarin	celecoxib	methazolamide	imatinib	chlorthalidone	sulfanilamide	acetaminophen	nilotinib	triethylenetetramine	dorzolamide	lacosamide	ethoxzolamide	valdecoxib	acetazolamide	dobutamine	phenol	quercetin	hydroquinone	sulpiride
CA13		brinzolamide	cianidanol	celecoxib	methazolamide	indapamide	sulfanilamide	topiramate	dorzolamide	lacosamide	ethoxzolamide	valdecoxib	acetazolamide	zonisamide	dobutamine	diclofenamide
CA6		brinzolamide	mafenide	cianidanol	coumarin	methazolamide	imatinib	chlorthalidone	trichlormethiazide	sulfanilamide	ethoxzolamide	valdecoxib	acetazolamide	zonisamide	diclofenamide	salicylic acid	celecoxib	sulthiame	indapamide	topiramate	nilotinib	triethylenetetramine	dorzolamide	lacosamide	dobutamine	furosemide	quercetin	sulpiride
GRIN2D		loperamide	procyclidine	phencyclidine	chlorpromazine	ketamine	orphenadrine	budipine	cycloserine	acamprosate	levorphanol	amantadine
GRIN3B		procyclidine	phencyclidine	chlorpromazine	ketamine	orphenadrine	budipine	cycloserine	acamprosate	levorphanol	amantadine
GRIN1		procyclidine	tacrine	memantine	budipine	acamprosate	levorphanol	amantadine	phencyclidine	chlorpromazine	ketamine	pentamidine	orphenadrine	cycloserine	ifenprodil
GRIN2A		procyclidine	tacrine	memantine	budipine	acamprosate	levorphanol	amantadine	felbamate	loperamide	phencyclidine	chlorpromazine	ketamine	pentamidine	orphenadrine	cycloserine	milnacipran
GRIN2B		procyclidine	tacrine	memantine	budipine	acamprosate	levorphanol	amantadine	felbamate	loperamide	phencyclidine	chlorpromazine	ketamine	orphenadrine	cycloserine	ifenprodil
GRIN2C		loperamide	procyclidine	phencyclidine	chlorpromazine	ketamine	orphenadrine	budipine	cycloserine	acamprosate	dextromethorphan	levorphanol	amantadine
GRIN3A		procaine	procyclidine	meperidine	riluzole	memantine	budipine	profenamine	dextropropoxyphene	ethanol	acamprosate	dextromethorphan	levorphanol	amantadine	phencyclidine	gabapentin	chlorpromazine	ketamine	ketobemidone	orphenadrine	cycloserine	methadone
EDNRA		exisulind	irbesartan	sulfisoxazole	ambrisentan	amiodarone	bosentan	macitentan	sulfathiazole
HRH4		amitriptyline	histamine	delavirdine	cinnarizine	thioridazine	zotepine	mianserin	pheniramine	chlorpheniramine	promethazine	sulfisoxazole	cyproheptadine	chlorpromazine	clozapine	loxapine	astemizole	mebhydrolin	paliperidone	diphenhydramine	doxepin
GPR35		nedocromil	lodoxamide	niflumic acid	bumetanide	tolcapone	dicoumarol	entacapone	furosemide	quercetin	cromoglicic acid
VKORC1		phenindione	ethyl biscoumacetate	dicoumarol	warfarin	phenprocoumon	acenocoumarol
CACNA1D		felodipine	manidipine	nifedipine	lacidipine	aranidipine	clevidipine	nimodipine	efonidipine	barnidipine	amlodipine	cilnidipine	isradipine	nisoldipine	dexniguldipine	levamlodipine	nitrendipine	nicardipine	azelnidipine	nilvadipine	bepridil	benidipine	lercanidipine
CACNA1C		nifedipine	aranidipine	nimodipine	verapamil	efonidipine	barnidipine	nisoldipine	drotaverine	levamlodipine	nicardipine	azelnidipine	lercanidipine	felodipine	manidipine	lacidipine	diltiazem	hydralazine	clevidipine	endralazine	amlodipine	cilnidipine	isradipine	cadralazine	dexniguldipine	mibefradil	nitrendipine	propranolol	nilvadipine	bepridil	benidipine
CACNA1H		felodipine	nifedipine	diltiazem	nimodipine	verapamil	efonidipine	amlodipine	methsuximide	isradipine	perhexiline	nisoldipine	dexniguldipine	mibefradil	nitrendipine	phensuximide	paramethadione	amiodarone	flunarizine	nicardipine	bepridil	benidipine
TOP2A		mitoxantrone	intoplicine	teniposide	valrubicin	idarubicin	etoposide	doxorubicin	ciprofloxacin	daunorubicin	amsacrine
TOP1		irinotecan	ribavirin	intoplicine	oleic acid	doxorubicin	belotecan	topotecan	yohimbine	amsacrine
ALPL		levamisole	theophylline	amifostine	miconazole	sulconazole
F10		nafamostat	ximelagatran	dabigatran etexilate	argatroban	apixaban	rivaroxaban	edoxaban
THRA		dextrothyroxine	amiodarone	dronedarone	liothyronine	levothyroxine	tiratricol
GABRA2		zaleplon	loprazolam	fospropofol	norfloxacin	etizolam	metharbital	estazolam	flunitrazepam	meprobamate	zolpidem	hexobarbital	pentobarbital	thiamylal	delorazepam	quazepam	sevoflurane	etomidate	thiocolchicoside	alfaxalone	methoxyflurane	adinazolam	alprazolam	talbutal	triclofos	isoflurane	diazepam	eszopiclone	propofol	desflurane	triazolam	chlordiazepoxide	halazepam	ofloxacin	methaqualone	clonazepam	halothane	liothyronine	progabide	flumazenil
GABRA3		loprazolam	zopiclone	fospropofol	norfloxacin	etizolam	metharbital	estazolam	flunitrazepam	meprobamate	zolpidem	hexobarbital	thiamylal	delorazepam	quazepam	sevoflurane	methoxyflurane	adinazolam	alprazolam	talbutal	triclofos	isoflurane	diazepam	eszopiclone	desflurane	triazolam	chlordiazepoxide	halazepam	methaqualone	clonazepam	midazolam	halothane	liothyronine	progabide	flumazenil
GABRA4		adinazolam	talbutal	triclofos	isoflurane	eszopiclone	desflurane	fospropofol	norfloxacin	metharbital	triazolam	ethanol	halazepam	methaqualone	clonazepam	thiamylal	delorazepam	sevoflurane	halothane	liothyronine	progabide	flumazenil	methoxyflurane
GABRA5		loprazolam	zopiclone	fospropofol	norfloxacin	etizolam	metharbital	estazolam	flunitrazepam	meprobamate	hexobarbital	thiamylal	delorazepam	sevoflurane	methoxyflurane	adinazolam	alprazolam	talbutal	triclofos	isoflurane	diazepam	eszopiclone	desflurane	triazolam	chlordiazepoxide	halazepam	methaqualone	clonazepam	midazolam	halothane	liothyronine	progabide	flumazenil
GABRA6		adinazolam	talbutal	triclofos	isoflurane	desflurane	fospropofol	norfloxacin	metharbital	triazolam	halazepam	lindane	methaqualone	clonazepam	thiamylal	delorazepam	sevoflurane	halothane	liothyronine	progabide	flumazenil	methoxyflurane
GABRB1		adinazolam	talbutal	triclofos	isoflurane	desflurane	fospropofol	metharbital	triazolam	halazepam	lindane	clonazepam	thiamylal	delorazepam	quazepam	sevoflurane	halothane	liothyronine	progabide	thiocolchicoside	flumazenil	methoxyflurane
GABRD		adinazolam	talbutal	triclofos	isoflurane	desflurane	fospropofol	metharbital	triazolam	ethanol	halazepam	methaqualone	clonazepam	thiamylal	delorazepam	sevoflurane	halothane	liothyronine	progabide	flumazenil	methoxyflurane
GABRE		talbutal	triclofos	isoflurane	desflurane	metharbital	halazepam	clonazepam	thiamylal	delorazepam	sevoflurane	halothane	liothyronine	progabide	flumazenil	methoxyflurane
GABRG1		adinazolam	talbutal	triclofos	isoflurane	desflurane	fospropofol	metharbital	triazolam	halazepam	clonazepam	thiamylal	delorazepam	sevoflurane	halothane	liothyronine	progabide	flumazenil	methoxyflurane
GABRG3		adinazolam	talbutal	triclofos	isoflurane	diazepam	eszopiclone	zopiclone	desflurane	fospropofol	metharbital	triazolam	halazepam	flunitrazepam	clonazepam	midazolam	thiamylal	delorazepam	sevoflurane	halothane	liothyronine	progabide	flumazenil	methoxyflurane
GABRP		talbutal	triclofos	isoflurane	desflurane	metharbital	halazepam	clonazepam	thiamylal	delorazepam	sevoflurane	halothane	liothyronine	progabide	flumazenil	methoxyflurane
GABRQ		talbutal	triclofos	isoflurane	desflurane	metharbital	halazepam	clonazepam	thiamylal	delorazepam	sevoflurane	halothane	liothyronine	progabide	flumazenil	methoxyflurane
THRB		dextrothyroxine	amiodarone	liothyronine	levothyroxine	tiratricol
HCN4		aprindine	quinidine	flecainide	verapamil	cibenzoline	lidocaine	disopyramide	propafenone	propranolol	amiodarone	ivabradine	dronedarone	mexiletine	bepridil
SCN10A		benzocaine	cinchocaine	procaine	ethotoin	ropivacaine	proparacaine	lamotrigine	tocainide	eslicarbazepine acetate	chloroprocaine	lidocaine	ambroxol	dyclonine	mephenytoin	oxybuprocaine	procainamide	rufinamide	phenazopyridine	orphenadrine	mexiletine
FDPS		alendronic acid	neridronic acid	minodronic acid	risedronic acid	zoledronic acid	pamidronic acid	incadronic acid	ibandronate
GAA		acarbose	miglustat	voglibose	migalastat	miglitol
PTGFR		latanoprost	enprostil	dinoprostone	misoprostol	iloprost	laropiprant	bimatoprost	dinoprost	travoprost	sulprostone	tafluprost
PTGER3		treprostinil	misoprostol	iloprost	laropiprant	dinoprost	travoprost	sulprostone	beraprost	latanoprost	enprostil	alprostadil	dinoprostone	mezlocillin	paliperidone
CYP11B1		metyrapone	letrozole	mitotane	ketoconazole	etomidate
PGR		dexamethasone	etonogestrel	dydrogesterone	levonorgestrel	megestrol acetate	triamcinolone	norethisterone	norethynodrel	norgestimate	fluticasone propionate	medroxyprogesterone acetate	norelgestromin	ethynodiol diacetate	tibolone	cyproterone acetate	mometasone furoate	fulvestrant	hydroxyprogesterone caproate	progesterone	promegestone	desogestrel	mifepristone	gestodene	spironolactone	dienogest	danazol	quingestanol acetate	drospirenone	tamoxifen
SHBG		estradiol benzoate	ethinylestradiol	testosterone	etonogestrel	gestrinone	androstenedione	levonorgestrel	cortisone acetate	estriol	norethisterone	hydrocortisone	medroxyprogesterone acetate	methyltestosterone	aldosterone	hydroxyprogesterone caproate	progesterone	prasterone	desogestrel	mesterolone	androstenediol	estrone	danazol	nandrolone	stanolone	estradiol
KCNA5		nifedipine	guanidine	quinidine	levobupivacaine	propafenone	bupivacaine	flecainide	dronedarone	dalfampridine	amifampridine	vernakalant
PTGER1		bupivacaine	treprostinil	iloprost	laropiprant	dinoprost	sulprostone	latanoprost	enprostil	alprostadil	levobupivacaine	dinoprostone	epoprostenol	limaprost	mezlocillin
PLG		nafamostat	ximelagatran	dabigatran etexilate	telaprevir	tranexamic acid	aminocaproic acid
CNR1		nabilone	orlistat	rimonabant	nimodipine	cefapirin	miconazole	mestranol	acetaminophen	flunarizine	dronabinol	palmidrol	mezlocillin	econazole
MAPK10		axitinib	nilotinib	sunitinib	afatinib	pazopanib	erlotinib	imatinib	nintedanib	gefitinib
ABL1		axitinib	sunitinib	erlotinib	ponatinib	sorafenib	imatinib	gefitinib	ceritinib	tofacitinib	lapatinib	radotinib	nilotinib	afatinib	dasatinib	crizotinib	pazopanib	vandetanib	mebendazole	nintedanib	ruxolitinib	bosutinib
FLT3		axitinib	sunitinib	palbociclib	erlotinib	ponatinib	sorafenib	imatinib	ruboxistaurin	gefitinib	cabozantinib	ceritinib	nilotinib	afatinib	dasatinib	crizotinib	pazopanib	vandetanib	nintedanib	quercetin	bosutinib
MAPK9		nilotinib	sunitinib	afatinib	erlotinib	sorafenib	imatinib	gefitinib
KDR		niclosamide	axitinib	sunitinib	erlotinib	ponatinib	sorafenib	lenvatinib	imatinib	regorafenib	gefitinib	vemurafenib	cabozantinib	ceritinib	dasatinib	pazopanib	vandetanib	mebendazole	nintedanib	quercetin	rivoceranib
MET		axitinib	sunitinib	erlotinib	gefitinib	cabozantinib	ceritinib	afatinib	crizotinib	pazopanib	vandetanib	nintedanib	quercetin	bosutinib
CSNK1E		sunitinib	afatinib	dasatinib	erlotinib	vandetanib	nintedanib	gefitinib	bosutinib
RIPK2		axitinib	afatinib	dasatinib	crizotinib	pazopanib	erlotinib	sorafenib	vandetanib	gefitinib	bosutinib	lapatinib
EPHB4		nilotinib	sunitinib	dasatinib	crizotinib	erlotinib	sorafenib	vandetanib	imatinib	nintedanib	gefitinib	bosutinib
GAK		axitinib	sunitinib	afatinib	dasatinib	pazopanib	erlotinib	vandetanib	imatinib	ruboxistaurin	ruxolitinib	gefitinib	bosutinib
SBK1		sunitinib	afatinib	dasatinib	crizotinib	erlotinib	nintedanib	ruxolitinib	gefitinib
MAP2K5		axitinib	sunitinib	erlotinib	sorafenib	ruboxistaurin	gefitinib	lapatinib	nilotinib	afatinib	dasatinib	pazopanib	vandetanib	nintedanib	bosutinib
CSNK1D		sunitinib	erlotinib	nintedanib	gefitinib	bosutinib
PRKD1		sunitinib	crizotinib	suramin	ingenol mebutate	nintedanib	gefitinib
EPHA1		nilotinib	dasatinib	crizotinib	sorafenib	vandetanib	nintedanib	gefitinib	bosutinib
MKNK1		sunitinib	afatinib	erlotinib	sorafenib	vandetanib	ruboxistaurin	gefitinib
FGR		axitinib	sunitinib	erlotinib	sorafenib	imatinib	gefitinib	ceritinib	nilotinib	dasatinib	crizotinib	ibrutinib	pazopanib	vandetanib	nintedanib	bosutinib
FRK		sunitinib	erlotinib	sorafenib	imatinib	gefitinib	nilotinib	afatinib	dasatinib	crizotinib	pazopanib	vandetanib	nintedanib	bosutinib
EPHA8		nilotinib	dasatinib	crizotinib	erlotinib	sorafenib	vandetanib	imatinib	gefitinib	bosutinib
EPHA3		nilotinib	sunitinib	dasatinib	crizotinib	erlotinib	sorafenib	vandetanib	nintedanib	ruxolitinib	gefitinib	bosutinib
STK10		axitinib	sunitinib	erlotinib	sorafenib	ruboxistaurin	gefitinib	lapatinib	nilotinib	afatinib	dasatinib	crizotinib	pazopanib	vandetanib	nintedanib	bosutinib
STK17B		sunitinib	erlotinib	nintedanib	ruxolitinib	gefitinib
HCK		sunitinib	erlotinib	sorafenib	ruboxistaurin	gefitinib	nilotinib	afatinib	dasatinib	ibrutinib	pazopanib	vandetanib	nintedanib	bosutinib
PHKG2		sunitinib	afatinib	vandetanib	nintedanib	ruxolitinib	gefitinib	bosutinib
CIT		sunitinib	afatinib	erlotinib	sorafenib	vandetanib	ruboxistaurin	gefitinib	bosutinib
HIPK4		sunitinib	afatinib	crizotinib	erlotinib	sorafenib	imatinib	nintedanib	gefitinib	bosutinib
MINK1		axitinib	sunitinib	dasatinib	crizotinib	erlotinib	vandetanib	nintedanib	ruboxistaurin	gefitinib	bosutinib
PIP4K2C		nilotinib	pazopanib	erlotinib	imatinib	gefitinib
IRAK4		sunitinib	crizotinib	vandetanib	nintedanib	gefitinib	bosutinib
STK36		dasatinib	pazopanib	erlotinib	sorafenib	gefitinib	bosutinib
KIT		niclosamide	axitinib	sunitinib	erlotinib	ponatinib	sorafenib	lenvatinib	imatinib	ruboxistaurin	gefitinib	cabozantinib	ceritinib	nilotinib	dasatinib	crizotinib	pazopanib	vandetanib	nintedanib	ruxolitinib	bosutinib	rivoceranib
ERBB4		afatinib	dasatinib	ibrutinib	erlotinib	vandetanib	gefitinib	bosutinib	lapatinib
STK17A		sunitinib	afatinib	erlotinib	imatinib	nintedanib	ruxolitinib	gefitinib
EPHA6		nilotinib	sunitinib	afatinib	dasatinib	crizotinib	erlotinib	sorafenib	vandetanib	nintedanib	gefitinib	bosutinib
TNIK		axitinib	sunitinib	dasatinib	pazopanib	erlotinib	sorafenib	vandetanib	nintedanib	ruboxistaurin	gefitinib	bosutinib
RPS6KA4		sunitinib	erlotinib	nintedanib	ruboxistaurin	ruxolitinib	gefitinib
SLK		axitinib	sunitinib	erlotinib	sorafenib	ruboxistaurin	gefitinib	lapatinib	afatinib	dasatinib	crizotinib	pazopanib	vandetanib	nintedanib	bosutinib
MKNK2		sunitinib	afatinib	erlotinib	sorafenib	vandetanib	ruxolitinib	gefitinib	ceritinib	tofacitinib
IRAK1		axitinib	sunitinib	afatinib	crizotinib	pazopanib	vandetanib	imatinib	nintedanib	ruxolitinib	gefitinib	bosutinib
LYN		niclosamide	sunitinib	erlotinib	ponatinib	sorafenib	imatinib	gefitinib	ceritinib	nilotinib	dasatinib	crizotinib	ibrutinib	pazopanib	vandetanib	nintedanib	bosutinib
EPHA5		nilotinib	sunitinib	dasatinib	crizotinib	erlotinib	sorafenib	vandetanib	gefitinib	bosutinib
PHKG1		sunitinib	afatinib	vandetanib	nintedanib	ruboxistaurin	ruxolitinib	gefitinib	bosutinib
EPHB1		nilotinib	sunitinib	dasatinib	crizotinib	erlotinib	sorafenib	vandetanib	imatinib	nintedanib	gefitinib	bosutinib
IRAK3		sunitinib	crizotinib	pazopanib	nintedanib	gefitinib
MAP3K2		sunitinib	dasatinib	crizotinib	pazopanib	erlotinib	nintedanib	ruboxistaurin	ruxolitinib	gefitinib	bosutinib
ABL2		axitinib	sunitinib	erlotinib	sorafenib	imatinib	gefitinib	nilotinib	dasatinib	crizotinib	pazopanib	vandetanib	nintedanib	bosutinib
BLK		axitinib	sunitinib	erlotinib	imatinib	gefitinib	nilotinib	afatinib	dasatinib	crizotinib	ibrutinib	pazopanib	vandetanib	nintedanib	bosutinib
ERBB3		afatinib	dasatinib	erlotinib	vandetanib	gefitinib	bosutinib	lapatinib
EPHB6		axitinib	sunitinib	erlotinib	sorafenib	gefitinib	nilotinib	afatinib	dasatinib	crizotinib	pazopanib	vandetanib	nintedanib	ruxolitinib	bosutinib
SIK2		sunitinib	dasatinib	crizotinib	pazopanib	erlotinib	vandetanib	nintedanib	gefitinib	bosutinib
CDK7		sunitinib	crizotinib	sorafenib	vandetanib	nintedanib	ruboxistaurin	ruxolitinib	gefitinib	bosutinib
DAPK3		sunitinib	erlotinib	nintedanib	ruboxistaurin	ruxolitinib	gefitinib
DCLK3		sunitinib	nintedanib	ruxolitinib	gefitinib	tofacitinib	bosutinib
RET		amitriptyline	axitinib	nortriptyline	sunitinib	erlotinib	ponatinib	sorafenib	amitriptylinoxide	lenvatinib	cyclobenzaprine	gefitinib	cabozantinib	ceritinib	tofacitinib	nilotinib	dasatinib	crizotinib	ibrutinib	pazopanib	vandetanib	nintedanib	ruxolitinib	bosutinib	rivoceranib
DMPK		dasatinib	crizotinib	erlotinib	ruboxistaurin	ruxolitinib	gefitinib	tofacitinib	bosutinib
MYLK2		axitinib	sunitinib	dasatinib	pazopanib	erlotinib	sorafenib	nintedanib	gefitinib
LTK		sunitinib	crizotinib	pazopanib	erlotinib	vandetanib	nintedanib	ruxolitinib	gefitinib	bosutinib
MAP3K19		axitinib	sunitinib	erlotinib	sorafenib	ruboxistaurin	gefitinib	dasatinib	crizotinib	pazopanib	vandetanib	nintedanib	ruxolitinib	bosutinib
AXL		axitinib	sunitinib	afatinib	crizotinib	erlotinib	sorafenib	vandetanib	nintedanib	quercetin	gefitinib	bosutinib
NUAK2		axitinib	sunitinib	crizotinib	nintedanib	ruboxistaurin	ruxolitinib	gefitinib	tofacitinib	bosutinib
TXK		axitinib	afatinib	dasatinib	crizotinib	ibrutinib	pazopanib	erlotinib	vandetanib	nintedanib	gefitinib	bosutinib
MAP3K3		axitinib	sunitinib	dasatinib	crizotinib	erlotinib	nintedanib	ruboxistaurin	ruxolitinib	gefitinib	bosutinib
CHEK2		sunitinib	ruboxistaurin	irofulven	gefitinib	bosutinib
NLK		dasatinib	pazopanib	sorafenib	gefitinib	bosutinib
NTRK1		amitriptyline	axitinib	sunitinib	crizotinib	sorafenib	nintedanib	ruxolitinib	ceritinib	bosutinib
COMT		cefotetan	opicapone	tolcapone	entacapone	dobutamine
PTGER2		rofecoxib	alprostadil	etoricoxib	treprostinil	dinoprostone	misoprostol	iloprost	laropiprant	dinoprost	mezlocillin	indomethacin
PTGDR2		dinoprostone	laropiprant	dinoprost	ramatroban	mezlocillin	fentiazac	indomethacin
AKR1C3		mefenamic acid	naproxen	diclofenac	flurbiprofen	tolfenamic acid	dexibuprofen	medroxyprogesterone acetate	ibuprofen	flufenamic acid	mezlocillin	meclofenamic acid	indomethacin
CXCL8		diclofenac	tolmetin	ibuprofen	mezlocillin	indomethacin
AKR1C2		mefenamic acid	naproxen	flurbiprofen	dexibuprofen	ursodeoxycholic acid	medroxyprogesterone acetate	flufenamic acid	meclofenamic acid	indomethacin
GLO1		sulindac	sulfamethazine	tolmetin	quercetin	acemetacin	indomethacin
KCNA7		guanidine	quinidine	amiodarone	flecainide	verapamil	dalfampridine	amifampridine	indomethacin
CYP3A5		isoniazid	ethambutol	pyrazinamide	cefapirin	cobicistat	gestodene
DPP4		linagliptin	beta-sitosterol	metformin	saxagliptin	omarigliptin	anagliptin	sitagliptin	teneligliptin	vildagliptin	alogliptin	gemigliptin	quercetin	trelagliptin
SLC22A3		famotidine	irinotecan	mitoxantrone	ondansetron	pentamidine	imatinib	metformin	chlorhexidine	bithionol
GFER		olanzapine	promethazine	thiethylperazine	alimemazine	chlorpromazine	phenelzine	dopamine	fenoldopam	promazine
IL5		dexamethasone	budesonide	tacrolimus	beclomethasone dipropionate	pimecrolimus
TEK		niclosamide	axitinib	sorafenib	cabozantinib	loperamide	nilotinib	crizotinib	pazopanib	cetirizine	vandetanib	nintedanib	ampicillin	bosutinib
CACNG1		nitrendipine	diltiazem	nimodipine	dronedarone	amlodipine	nilvadipine	buflomedil	desipramine
CACNA1G		mibefradil	phensuximide	trimethadione	paramethadione	flunarizine	zonisamide	methsuximide	ethosuximide	levetiracetam	pimozide	perhexiline
ABCC4		irinotecan	tioguanine	mercaptopurine	methotrexate	azathioprine	topotecan
KCNMA1		bendroflumethiazide	hydrochlorothiazide	pinacidil	benzthiazide	estradiol	chlorzoxazone
HBA1		primaquine	quinine	hydroxychloroquine	nomifensine	mefloquine
AURKA		niclosamide	axitinib	sunitinib	dasatinib	crizotinib	pazopanib	erlotinib	sorafenib	doxorubicin	sulfadiazine
TUBB		paclitaxel	vinorelbine	docetaxel	eribulin	vinblastine	colchicine	cabazitaxel	vincristine	ixabepilone	podofilox	vinflunine
TUBB1		paclitaxel	vinorelbine	docetaxel	eribulin	vinblastine	cabazitaxel	vincristine	ixabepilone	podofilox	vinflunine
TUBB2A		paclitaxel	vinorelbine	docetaxel	eribulin	vinblastine	cabazitaxel	vincristine	ixabepilone	podofilox	vinflunine
TUBB2B		paclitaxel	vinorelbine	docetaxel	eribulin	vinblastine	cabazitaxel	vincristine	ixabepilone	podofilox	vinflunine
TUBB3		paclitaxel	vinorelbine	docetaxel	eribulin	vinblastine	cabazitaxel	vincristine	ixabepilone	podofilox	vinflunine
TUBB4A		paclitaxel	vinorelbine	docetaxel	eribulin	vinblastine	cabazitaxel	vincristine	ixabepilone	podofilox	vinflunine
TUBB4B		paclitaxel	vinorelbine	docetaxel	eribulin	vinblastine	colchicine	cabazitaxel	anhydrovinblastine	vincristine	ixabepilone	podofilox	vinflunine
TUBB6		paclitaxel	vinorelbine	docetaxel	eribulin	vinblastine	cabazitaxel	vincristine	ixabepilone	podofilox	vinflunine
TUBB8		paclitaxel	vinorelbine	docetaxel	eribulin	vinblastine	cabazitaxel	vincristine	ixabepilone	podofilox	vinflunine
PTGIR		enprostil	selexipag	alprostadil	treprostinil	dinoprostone	iloprost	laropiprant	epoprostenol	beraprost
PTGER4		enprostil	alprostadil	treprostinil	dinoprostone	misoprostol	iloprost	epoprostenol	dinoprost	sulprostone	mezlocillin	beraprost
PTGDR		alprostadil	treprostinil	dinoprostone	iloprost	laropiprant	dinoprost	ramatroban	mezlocillin
SCN4B		quinidine	propafenone	encainide	mexiletine	hydroquinidine	lorcainide
SCN3B		quinidine	propafenone	encainide	mexiletine	hydroquinidine	lorcainide
SCN2B		quinidine	propafenone	encainide	mexiletine	hydroquinidine	lorcainide
SCN1B		quinidine	propafenone	encainide	mexiletine	hydroquinidine	lorcainide
BCHE		promethazine	tacrine	quinidine	rivastigmine	neostigmine	profenamine	quercetin	bambuterol	donepezil	physostigmine	galantamine	pyridostigmine
STAT3		niclosamide	ouabain	digoxin	nifuroxazide	digitoxin
NR3C2		desoxycorticosterone pivalate	dexamethasone	aldosterone	nimodipine	progesterone	eplerenone	desoxycorticosterone acetate	mifepristone	spironolactone	prednisolone	medroxyprogesterone acetate	drospirenone	canrenone
FABP2		bezafibrate	flurbiprofen	progesterone	fenofibric acid	meclofenamic acid
SERPINA6		aldosterone	hydroxyprogesterone caproate	testosterone	progesterone	prasterone	hydrocortisone acetate	androstenedione	cortisone acetate	androstenediol	prednisolone	estriol	estrone	hydrocortisone	nandrolone	stanolone	estradiol
CDKL2		axitinib	sunitinib	crizotinib	sorafenib	nintedanib
FLT1		axitinib	sunitinib	dasatinib	crizotinib	pazopanib	erlotinib	sorafenib	lenvatinib	vandetanib	nintedanib
FGFR3		axitinib	sunitinib	dasatinib	crizotinib	pazopanib	sorafenib	vandetanib	nintedanib	ceritinib
INSR		nilotinib	sunitinib	crizotinib	sorafenib	osimertinib	imatinib	nintedanib	ceritinib	lapatinib
PDGFRA		axitinib	sunitinib	erlotinib	ponatinib	sorafenib	lenvatinib	imatinib	ceritinib	nilotinib	dasatinib	pazopanib	vandetanib	nintedanib	bosutinib
RPS6KA6		sunitinib	afatinib	sorafenib	vandetanib	nintedanib	ruboxistaurin	ruxolitinib	tofacitinib	bosutinib
MAP3K20		axitinib	nilotinib	dasatinib	sorafenib	vandetanib	imatinib	bosutinib
HIPK3		sunitinib	sorafenib	nintedanib	ruboxistaurin	ruxolitinib	bosutinib
HIPK2		sunitinib	sorafenib	nintedanib	ruboxistaurin	ruxolitinib	bosutinib
RAF1		nilotinib	dasatinib	pazopanib	sorafenib	imatinib	dabrafenib	vemurafenib
MAP4K1		axitinib	nilotinib	sunitinib	dasatinib	crizotinib	pazopanib	sorafenib	vandetanib	nintedanib	ruboxistaurin	bosutinib
BRAF		nilotinib	dasatinib	pazopanib	sorafenib	imatinib	regorafenib	dabrafenib	ruxolitinib	vemurafenib
MAP3K7		sunitinib	dasatinib	crizotinib	sorafenib	nintedanib	ruxolitinib	bosutinib
CLK1		nilotinib	sunitinib	sorafenib	imatinib	nintedanib	ruboxistaurin	bosutinib
HIPK1		sunitinib	sorafenib	nintedanib	ruboxistaurin	ruxolitinib	bosutinib
TTK		axitinib	sunitinib	pazopanib	erlotinib	sorafenib	nintedanib	ruxolitinib
EPHA2		nilotinib	dasatinib	crizotinib	sorafenib	vandetanib	nintedanib	bosutinib
PLK4		axitinib	sunitinib	crizotinib	pazopanib	erlotinib	sorafenib	vandetanib	imatinib	nintedanib	ruboxistaurin	ruxolitinib
JAK3		axitinib	sunitinib	palbociclib	erlotinib	sorafenib	ruboxistaurin	baricitinib	ceritinib	tofacitinib	dasatinib	crizotinib	ibrutinib	pazopanib	nintedanib	ruxolitinib	bosutinib
CSK		axitinib	nilotinib	dasatinib	erlotinib	ponatinib	sorafenib	vandetanib	bosutinib	rivoceranib
TAOK1		nilotinib	sunitinib	crizotinib	pazopanib	sorafenib	ruboxistaurin	ruxolitinib	bosutinib
TNNI3K		nilotinib	dasatinib	crizotinib	erlotinib	sorafenib	vandetanib	imatinib	bosutinib
AURKC		axitinib	sunitinib	crizotinib	pazopanib	erlotinib	sorafenib	vandetanib	nintedanib	ruboxistaurin	ruxolitinib
PDGFRB		axitinib	sunitinib	erlotinib	sorafenib	lenvatinib	imatinib	ruboxistaurin	lapatinib	nilotinib	dasatinib	pazopanib	vandetanib	nintedanib	bosutinib
FGFR1		niclosamide	axitinib	sunitinib	ponatinib	sorafenib	lenvatinib	imatinib	ruboxistaurin	nilotinib	dasatinib	pazopanib	vandetanib	nintedanib
FGFR2		axitinib	nilotinib	sunitinib	dasatinib	ibrutinib	pazopanib	erlotinib	sorafenib	vandetanib	imatinib	nintedanib	ceritinib
MAP4K5		axitinib	sunitinib	dasatinib	crizotinib	pazopanib	sorafenib	vandetanib	nintedanib	ruboxistaurin	bosutinib
AURKB		axitinib	sunitinib	dasatinib	crizotinib	erlotinib	sorafenib	nintedanib	quercetin
EPHA7		sunitinib	crizotinib	erlotinib	sorafenib	vandetanib
TAOK2		dasatinib	crizotinib	pazopanib	sorafenib	ruboxistaurin	ruxolitinib	bosutinib
EPHA4		nilotinib	dasatinib	crizotinib	sorafenib	vandetanib	bosutinib
NTRK3		nilotinib	sunitinib	crizotinib	sorafenib	nintedanib	ruxolitinib	bosutinib
CDK2		palbociclib	sorafenib	nintedanib	quercetin	ceritinib	lapatinib
EPHX2		fulvestrant	sorafenib	regorafenib	rutin	quercetin	zileuton	triclocarban
TAOK3		nilotinib	sunitinib	dasatinib	crizotinib	pazopanib	sorafenib	ruboxistaurin	ruxolitinib	bosutinib
SRMS		dasatinib	pazopanib	sorafenib	vandetanib	bosutinib
CSF1R		axitinib	nilotinib	sunitinib	dasatinib	crizotinib	pazopanib	sorafenib	vandetanib	imatinib	nintedanib	bosutinib
FLT4		axitinib	sunitinib	pazopanib	erlotinib	sorafenib	lenvatinib	vandetanib	nintedanib
DDR2		axitinib	nilotinib	sunitinib	dasatinib	pazopanib	sorafenib	vandetanib	imatinib	nintedanib	bosutinib	dactinomycin
TIE1		axitinib	nilotinib	sunitinib	crizotinib	pazopanib	erlotinib	sorafenib	vandetanib	nintedanib	bosutinib
DDR1		axitinib	nilotinib	sunitinib	dasatinib	crizotinib	pazopanib	erlotinib	sorafenib	vandetanib	imatinib	nintedanib	bosutinib
MAP4K4		axitinib	sunitinib	dasatinib	pazopanib	sorafenib	vandetanib	nintedanib	bosutinib
NTRK2		nilotinib	sunitinib	crizotinib	sorafenib	nintedanib	ruxolitinib	ceritinib	bosutinib
EPHB2		nilotinib	dasatinib	sorafenib	vandetanib	bosutinib
STK33		sunitinib	sorafenib	vandetanib	nintedanib	ruboxistaurin	bosutinib
MERTK		axitinib	sunitinib	crizotinib	pazopanib	erlotinib	sorafenib	vandetanib	nintedanib	bosutinib
TNK1		axitinib	sunitinib	crizotinib	pazopanib	erlotinib	sorafenib	nintedanib	tofacitinib
CCKAR		paclitaxel	sincalide	ceruletide	dexloxiglumide	chlordiazepoxide
PRNP		chloroquine	promethazine	quinacrine	chlortetracycline	chlorpromazine	imipramine	acepromazine	promazine
CALM1		haloperidol	loperamide	aprindine	cyproheptadine	chlorpromazine	domperidone	quercetin	trifluoperazine	astemizole	pimozide
GUCY1A2		isosorbide mononitrate	benzydamine	nitroglycerin	nitric oxide	isosorbide dinitrate
GUCY1A1		isosorbide mononitrate	benzydamine	nitroglycerin	nitric oxide	isosorbide dinitrate
GUCY1B2		isosorbide mononitrate	benzydamine	nitroglycerin	nitric oxide	isosorbide dinitrate
GUCY1B1		isosorbide mononitrate	benzydamine	nitroglycerin	nitric oxide	isosorbide dinitrate	riociguat
ANXA1		cortisone acetate	prednisolone	betamethasone	triamcinolone	dexamethasone	clobetasol propionate	hydrocortisone	methylprednisolone	desoximetasone	prednisone
MMP1		irinotecan	aminoquinuride	cefotetan	nimesulide	doxazosin	prazosin	sulfasalazine	cefapirin
NQO2		chloroquine	dabigatran etexilate	primaquine	terazosin	bunazosin	imatinib	prazosin	melatonin
SLC29A4		dipyridamole	fluoxetine	quinidine	quinine	verapamil	desipramine
CNR2		nabilone	rimonabant	dronabinol	palmidrol	mezlocillin
HRH3		histamine	fluoxetine	ofloxacin	pitolisant	azelastine	betahistine	decamethonium	donepezil
MC4R		afamelanotide	amiodarone	chlorpromazine	miconazole	astemizole	tetracosactide	tamoxifen
MC5R		paclitaxel	afamelanotide	amiodarone	chlorpromazine	miconazole	astemizole	econazole	sertraline	fluphenazine	tamoxifen
MC3R		afamelanotide	amiodarone	chlorpromazine	miconazole	astemizole	econazole	tamoxifen
EBP		haloperidol	opipramol	amiodarone	clomifene	raloxifene	trifluoperazine	buflomedil	naftifine	trifluperidol	tamoxifen
PDPK1		niclosamide	sunitinib	celecoxib	nintedanib	ruboxistaurin
GRK4		axitinib	sunitinib	crizotinib	erlotinib	nintedanib	ruboxistaurin	ruxolitinib	bosutinib
ULK3		axitinib	sunitinib	dasatinib	crizotinib	erlotinib	vandetanib	nintedanib	ruxolitinib	tofacitinib	bosutinib
DYRK2		sunitinib	afatinib	crizotinib	erlotinib	ruxolitinib
JAK2		niclosamide	axitinib	sunitinib	erlotinib	imatinib	baricitinib	ceritinib	tofacitinib	nilotinib	dasatinib	crizotinib	pazopanib	nintedanib	ruxolitinib	bosutinib
EIF2AK2		axitinib	sunitinib	crizotinib	pazopanib	erlotinib
TBK1		sunitinib	crizotinib	erlotinib	nintedanib	ruboxistaurin	ruxolitinib	bosutinib
AAK1		axitinib	sunitinib	crizotinib	pazopanib	erlotinib	nintedanib	ruboxistaurin	ruxolitinib	bosutinib
EIF2AK4		sunitinib	dasatinib	erlotinib	nintedanib	bosutinib
TYRO3		sunitinib	crizotinib	erlotinib	vandetanib	nintedanib	bosutinib
YES1		axitinib	nilotinib	sunitinib	dasatinib	crizotinib	ibrutinib	pazopanib	erlotinib	vandetanib	nintedanib	bosutinib
SRPK3		axitinib	sunitinib	crizotinib	erlotinib	nintedanib	ruboxistaurin	ruxolitinib	bosutinib
ALK		sunitinib	crizotinib	pazopanib	erlotinib	vandetanib	nintedanib	quercetin	ruxolitinib	ceritinib	bosutinib
LRRK2		axitinib	sunitinib	erlotinib	nintedanib	ruboxistaurin	ruxolitinib	tofacitinib	bosutinib
BMP2K		axitinib	sunitinib	crizotinib	pazopanib	erlotinib	nintedanib	ruboxistaurin	ruxolitinib	tofacitinib	bosutinib
CAMK2D		sunitinib	erlotinib	ruboxistaurin	ruxolitinib	tofacitinib
TYK2		axitinib	sunitinib	dasatinib	crizotinib	pazopanib	erlotinib	imatinib	nintedanib	ruxolitinib	baricitinib	tofacitinib	bosutinib
RIPK4		axitinib	sunitinib	crizotinib	erlotinib	vandetanib	nintedanib	ruxolitinib
SCN11A		benzocaine	ethotoin	mephenytoin	procainamide	rufinamide	tocainide	cocaine	eslicarbazepine acetate	phenazopyridine
SCN7A		benzocaine	ethotoin	mephenytoin	procainamide	rufinamide	tocainide	eslicarbazepine acetate	phenazopyridine
KCNA10		guanidine	verapamil	ketoconazole	dalfampridine	amifampridine	pimozide
KCNQ2		guanidine	dronedarone	linopirdine	ezogabine	flupirtine	dalfampridine	amifampridine
KCNQ3		guanidine	ezogabine	flupirtine	dalfampridine	amifampridine
KCNQ4		guanidine	linopirdine	ezogabine	dalfampridine	amifampridine	bepridil
KCNQ5		guanidine	linopirdine	ezogabine	dalfampridine	amifampridine
ABCC10		paclitaxel	docetaxel	vinblastine	anhydrovinblastine	vincristine
MPO		cadralazine	nimesulide	propylthiouracil	nomifensine	quercetin	flufenamic acid
NISCH		naphazoline	phentolamine	moxonidine	tizanidine	guanfacine	rilmenidine	fenoxazoline	oxymetazoline	clonidine	cefapirin	guanabenz	metizoline
AKR1B10		mefenamic acid	diclofenac	tolrestat	epalrestat	flufenamic acid	enoxolone
AKR1C1		mefenamic acid	medroxyprogesterone acetate	benzbromarone	flufenamic acid	meclofenamic acid
HTR4		metoclopramide	cisapride	prucalopride	tegaserod	tropisetron	mosapride	vilazodone
CACNA1I		mibefradil	phensuximide	paramethadione	flunarizine	methsuximide	pimozide	perhexiline
BMX		nilotinib	dasatinib	crizotinib	ibrutinib	imatinib	bosutinib
SYK		dasatinib	crizotinib	pazopanib	imatinib	quercetin	ceritinib	bosutinib
CLK4		nilotinib	sunitinib	imatinib	nintedanib	ruboxistaurin	ruxolitinib	bosutinib
MAPK8		axitinib	nilotinib	pazopanib	imatinib	nintedanib	ruxolitinib
BCR		nilotinib	dasatinib	ponatinib	imatinib	bosutinib
HSD11B1		acetoxolone	carbenoxolone	glycyrrhizic acid	furosemide	enoxolone
PRSS1		camostat	nafamostat	propamidine	dabigatran etexilate	pentamidine	sulfaguanidine	hexamidine
ST14		nafamostat	pentamidine	dibrompropamidine	hexamidine	rivaroxaban
GLRB		nifedipine	isoflurane	desflurane	halothane	tropisetron
MTNR1A		ramelteon	malathion	tasimelteon	dopamine	melatonin	agomelatine
BACE1		cianidanol	phloroglucinol	quercetin	tyramine	donepezil	hydroxyamphetamine
MTOR		dasatinib	everolimus	temsirolimus	sirolimus	tacrolimus	ridaforolimus
SLC6A1		tiagabine	cocaine	gamma-aminobutyric acid	stiripentol	alfaxalone
TBXA2R		tretoquinol	dinoprostone	iloprost	laropiprant	dinoprost	seratrodast	ramatroban
MTNR1B		ramelteon	tasimelteon	dopamine	melatonin	agomelatine
GSK3B		niclosamide	nintedanib	ruboxistaurin	quercetin	hesperetin
MYLK		nifedipine	sunitinib	fasudil	nintedanib	ruboxistaurin	ruxolitinib	bosutinib
BTK		sunitinib	dasatinib	crizotinib	ibrutinib	mitoxantrone	vandetanib	nintedanib	ceritinib	bosutinib
MAP2K1		axitinib	sunitinib	trametinib	dasatinib	vandetanib	nintedanib	ruxolitinib	cobimetinib	bosutinib
STK35		sunitinib	dasatinib	crizotinib	vandetanib	nintedanib	bosutinib
MAP3K13		sunitinib	dasatinib	crizotinib	nintedanib	bosutinib
MAP3K4		axitinib	sunitinib	dasatinib	vandetanib	bosutinib
BMPR1B		axitinib	sunitinib	dasatinib	crizotinib	pazopanib	vandetanib	ruxolitinib
STK4		axitinib	sunitinib	dasatinib	crizotinib	nintedanib	ruboxistaurin	bosutinib
NEK2		sunitinib	dasatinib	pazopanib	quercetin	bosutinib
TNK2		axitinib	sunitinib	dasatinib	crizotinib	nintedanib	ruxolitinib	bosutinib
MAP4K3		axitinib	sunitinib	dasatinib	crizotinib	pazopanib	vandetanib	nintedanib	ruboxistaurin	bosutinib
STK26		sunitinib	dasatinib	crizotinib	nintedanib	ruxolitinib	bosutinib
MAP2K2		axitinib	sunitinib	trametinib	dasatinib	vandetanib	nintedanib	ruxolitinib	cobimetinib	bosutinib
MAP4K2		axitinib	sunitinib	dasatinib	crizotinib	pazopanib	vandetanib	nintedanib	ruboxistaurin	ruxolitinib	tofacitinib	bosutinib
SIK1		axitinib	sunitinib	dasatinib	pazopanib	vandetanib	nintedanib	bosutinib
DPP8		sitagliptin	teneligliptin	vildagliptin	saxagliptin	anagliptin
DPP9		sitagliptin	teneligliptin	linagliptin	vildagliptin	gemigliptin	saxagliptin	anagliptin
PRKCQ		sunitinib	suramin	nintedanib	ruboxistaurin	bosutinib
DCLK1		sunitinib	crizotinib	nintedanib	ruxolitinib	tofacitinib
CAMK1		sunitinib	pazopanib	nintedanib	ruxolitinib	tofacitinib
FGFR4		sunitinib	pazopanib	vandetanib	nintedanib	ceritinib
SRPK1		axitinib	sunitinib	crizotinib	nintedanib	ruboxistaurin	ruxolitinib
RIOK3		axitinib	sunitinib	crizotinib	nintedanib	ruboxistaurin	ruxolitinib	bosutinib
MAP2K3		sunitinib	crizotinib	nintedanib	ruxolitinib	bosutinib
RPS6KA1		sunitinib	palbociclib	vandetanib	nintedanib	ruboxistaurin	ruxolitinib	tofacitinib
JAK1		sunitinib	crizotinib	nintedanib	ruxolitinib	baricitinib	ceritinib	tofacitinib
ITK		axitinib	sunitinib	crizotinib	ibrutinib	pazopanib	nintedanib	bosutinib
NUAK1		sunitinib	nintedanib	ruboxistaurin	quercetin	bosutinib
PRKD3		sunitinib	crizotinib	suramin	nintedanib	bosutinib
CLK2		sunitinib	nintedanib	ruboxistaurin	ruxolitinib	bosutinib
GRK7		sunitinib	nintedanib	ruboxistaurin	ruxolitinib	tofacitinib	bosutinib
FER		sunitinib	crizotinib	pazopanib	nintedanib	bosutinib
STK16		axitinib	sunitinib	pazopanib	nintedanib	ruxolitinib
RPS6KA5		sunitinib	fasudil	nintedanib	ruboxistaurin	ruxolitinib
CSNK2A2		axitinib	sunitinib	nintedanib	ruboxistaurin	ruxolitinib
PKN2		axitinib	sunitinib	fasudil	nintedanib	ruboxistaurin	tofacitinib	bosutinib
ROCK1		sunitinib	crizotinib	fasudil	ruxolitinib	ripasudil	tofacitinib	bosutinib
ANKK1		axitinib	sunitinib	crizotinib	ruxolitinib	bosutinib
CAMKK2		axitinib	sunitinib	crizotinib	nintedanib	ruboxistaurin	bosutinib
CAMK1D		sunitinib	nintedanib	ruboxistaurin	ruxolitinib	tofacitinib	bosutinib
STK3		axitinib	sunitinib	crizotinib	nintedanib	ruboxistaurin	tofacitinib	bosutinib
PRKAA1		sunitinib	crizotinib	vandetanib	nintedanib	bosutinib
RPS6KA2		sunitinib	nintedanib	ruboxistaurin	ruxolitinib	tofacitinib	bosutinib
ULK2		axitinib	sunitinib	crizotinib	nintedanib	ruxolitinib	bosutinib
CDK16		axitinib	sunitinib	pazopanib	nintedanib	ruboxistaurin	bosutinib
PTK2		sunitinib	crizotinib	nintedanib	quercetin	chloropyramine	bosutinib
CSNK2A1		sunitinib	nintedanib	ruboxistaurin	quercetin	ruxolitinib
CAMK2A		sunitinib	nintedanib	ruboxistaurin	ruxolitinib	tofacitinib	bosutinib
IKBKE		sunitinib	crizotinib	nintedanib	ruxolitinib	bosutinib
ROCK2		sunitinib	crizotinib	fasudil	vandetanib	ruxolitinib	ceritinib	ripasudil	tofacitinib	bosutinib
DYRK1A		sunitinib	afatinib	palbociclib	ruboxistaurin	ruxolitinib
FES		sunitinib	crizotinib	pazopanib	nintedanib	bosutinib
MAP3K9		axitinib	sunitinib	pazopanib	nintedanib	ruboxistaurin	bosutinib
MAP2K4		sunitinib	pazopanib	nintedanib	ruboxistaurin	ruxolitinib	bosutinib
MAP3K12		axitinib	sunitinib	crizotinib	nintedanib	bosutinib
RIPK1		axitinib	sunitinib	crizotinib	pazopanib	nintedanib
PIP5K1A		sunitinib	crizotinib	nintedanib	ruboxistaurin	bosutinib
RIOK1		axitinib	sunitinib	crizotinib	nintedanib	ruboxistaurin	ruxolitinib	bosutinib
CDK4		sunitinib	palbociclib	nintedanib	ribociclib	ruboxistaurin	quercetin	ceritinib
RPS6KB1		sunitinib	crizotinib	vandetanib	nintedanib	ruboxistaurin	bosutinib
ULK1		sunitinib	crizotinib	nintedanib	ruxolitinib	bosutinib
PKN1		sunitinib	fasudil	nintedanib	ruboxistaurin	quercetin	tofacitinib	bosutinib
PRKCA		sunitinib	suramin	ingenol mebutate	ruboxistaurin	dequalinium
GPBAR1		cholic acid	obeticholic acid	ursodeoxycholic acid	deoxycholic acid	chenodeoxycholic acid
HDAC10		vorinostat	romidepsin	bufexamac	bendamustine	panobinostat
HDAC8		phenylbutyric acid	vorinostat	romidepsin	bendamustine	panobinostat
PRKCD		suramin	ingenol mebutate	ruboxistaurin	tofacitinib	bosutinib
PRKCE		fasudil	suramin	ingenol mebutate	ruboxistaurin	ruxolitinib	bosutinib
SLC5A2		dapagliflozin	empagliflozin	tofogliflozin	canagliflozin	ipragliflozin	luseogliflozin
SLC5A1		dapagliflozin	empagliflozin	tofogliflozin	canagliflozin	ipragliflozin	luseogliflozin
ROS1		axitinib	crizotinib	pazopanib	nintedanib	ruboxistaurin	ceritinib
